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CHEMBL3099774 (CID 53495081) - Compound BioActivity Data
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BioActivity Outcomes:
Active(2)
 
 
Inactive(1)
 
 
Unspecified(1)
 
 
Top Targets:
7tm 4(3)
 
 
 
BioAssay Types:
Literature(2)
 
 
 
Confirmatory(2)
 
 
 
BioActivity Types:
EC50(3)
 
 
 
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 4    Data Row: 4   Total Pages: 1   
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#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID194166546]
EC50 9.4Agonist activity at NTR1 in human U2OS cells after 1 hr by beta-arrestin GFP reporter gene assay [AID1061686, Type: Literature]Neurotensin receptor type 1 [gi:62297312]
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2
[SID126723250]
EC50_Mean 9.41SAR analysis of small molecule Agonists NTR1 in a image based assay set 3 [AID602356, Type: confirmatory]neurotensin receptor type 1 [Homo sapiens] [gi:110611243]
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3
[SID194166546]
Agonist activity at NTR1 in human U2OS cells after 1 hr by beta-arrestin GFP reporter gene assay relative to NT peptide [AID1061685, Type: Literature]Neurotensin receptor type 1 [gi:62297312]
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4
[SID126723250]
EC50_Mean 80SAR analysis of small molecule NTR1 agonists in a image based NTR2 selectivity assay set 2 [AID602334, Type: confirmatory]neurotensin receptor type 2 [Homo sapiens] [gi:6912538]
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