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CHEMBL1818330 (CID 53465487) - Compound BioActivity Data
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BioActivity Outcomes:
Active(2)
 
 
Unspecified(2)
 
 
Top Targets:
7TM GPCR Srx(2)
 
 
BioAssay Types:
Literature(4)
 
 
 
BioActivity Types:
Ki(2)
 
 
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Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 4    Data Row: 4   Total Pages: 1   
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#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID134451430]
Ki 0.0022Displacement of [3H]diprenorphine from human kappa opioid receptor expressed in CHO cells after 1 hr by liquid scintillation counting [AID613641, Type: Literature]Kappa-type opioid receptor [gi:116242691]
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2
[SID134451430]
Ki 0.089Displacement of [3H]diprenorphine from human mu opioid receptor expressed in CHO cells after 1 hr by liquid scintillation counting [AID613642, Type: Literature]Mu-type opioid receptor [gi:2851402]
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3
[SID134451430]
Efflux ratio of permeability from basolateral to apical side over apical to basolateral side in MDCK cells expressing human MDR1 [AID613644, Type: Literature]
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4
[SID134451430]
Clearance in human liver microsomes [AID613645, Type: Literature]
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