4-Bromophenethylamine (CID 533915) - BioAssay Data Summary for Compound
.
BioActivity Outcomes:
Active(2)
 
 
Unspecified(1)
 
 
Top Targets:
7TM GPCR Srsx(2)
 
 
 
BioAssay Types:
Literature(3)
 
 
 
BioActivity Types:
EC50(1)
 
 
Ki(1)
 
 
SAR
Target summary
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 3    Data Row: 3   Total Pages: 1   
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#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID103623746]
EC50 1.54Agonist activity at human trace amine associated receptor 1 expressed in RD-HGA16 CHO-K1 cells coexpressed with Galpha16 protein assessed as internal calcium mobilization by calcium 3 assay [AID341210, Type: Literature]Trace amine-associated receptor 1 [gi:38258636]
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2
[SID103623746]
EC50 1.54Agonist activity at human trace amine associated receptor 1 expressed in RD-HGA16 CHO-K1 cells coexpressed with Galpha16 protein assessed as internal calcium mobilization by calcium 3 assay [AID341210, Type: Literature]Trace amine-associated receptor 1 [gi:38258636]
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3
[SID103623746]
Ki 1.77Displacement of [3H]ketanserin from 5HT2A receptor expressed in NIH3T3 cells [AID389734, Type: Literature]
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4
[SID103623746]
 Agonist activity at human trace amine associated receptor 1 expressed in RD-HGA16 CHO-K1 cells coexpressed with Galpha16 protein assessed as internal calcium mobilization by calcium 3 assay relative to 2-phenylethanamine [AID341211, Type: Literature]Trace amine-associated receptor 1 [gi:38258636]
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5
[SID103623746]
 Agonist activity at human trace amine associated receptor 1 expressed in RD-HGA16 CHO-K1 cells coexpressed with Galpha16 protein assessed as internal calcium mobilization by calcium 3 assay relative to 2-phenylethanamine [AID341211, Type: Literature]Trace amine-associated receptor 1 [gi:38258636]
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