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CHEMBL2203536 (CID 53377446) - Compound BioActivity Data
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BioActivity Outcomes:
Active(2)
 
 
Inconclusive(1)
 
 
Top Targets:
STKc STK33(2)
 
 
BioAssay Types:
Literature(2)
 
 
 
Confirmatory(1)
 
 
BioActivity Types:
IC50(2)
 
 
 
AC50(1)
 
 
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Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 3    Data Row: 3   Total Pages: 1   
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#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID125299423]
AC50_uM 1.54STK-33 Kinase Inhibition Measured in Biochemical System Using Plate Reader - 2052-02_Inhibitor_Dose_DryPowder_Activity_Set3 [AID602158, Type: confirmatory]serine/threonine-protein kinase 33 isoform a [Homo sapiens] [gi:23943882]
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2
[SID163339154]
IC50 1.6Inhibition of N-terminal 6His-tagged full length human recombinant STK33 using myelin basic protein as substrate incubated for 15 mins before initiation of kinase reaction measured after 1 hr by ADP-glo assay [AID712545, Type: Literature]Serine/threonine-protein kinase 33 [gi:74761329]
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3
[SID163339154]
IC50 Inhibition of His-tagged recombinant catalytic fragment of PKA assessed as phosphorylation of fluorescent-labeled peptide 21substrate by caliper capillary electrophoresis [AID712541, Type: Literature]
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