BRD-K66645150-001-01-4 (CID 53377419) - BioAssay Data Summary for Compound
.
BioActivity Outcomes:
Inactive(2)
 
 
Top Targets:
STKc AGC(1)
 
 
STKc PKA(1)
 
 
BioAssay Types:
Confirmatory(2)
 
 
BioActivity Types:
AC50(2)
 
 
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 2    Data Row: 2   Total Pages: 1   
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#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID125299379]
AC50 Protein Kinase A Activity Assay Measured in Biochemical System Using Plate Reader - 2052-04_Inhibitor_Dose_DryPowder_Activity_Set2 [AID588629, Type: confirmatory]cAMP-dependent protein kinase catalytic subunit alpha isoform 1 [Homo sapiens] [gi:4506055]
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2
[SID125299379]
AC50 Protein Kinase A Activity Assay Measured in Biochemical System Using Plate Reader - 2052-04_Inhibitor_Dose_DryPowder_Activity_Set2 [AID588629, Type: confirmatory]cAMP-dependent protein kinase catalytic subunit alpha isoform 1 [Homo sapiens] [gi:4506055]
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3
[SID125299379]
AC50 Counter screen for activity against Aurora B, in dose Measured in Biochemical System Using Scintillation - 2052-06_Inhibitor_Dose_DryPowder_Activity_Set3 [AID588808, Type: confirmatory]aurora kinase B [Homo sapiens] [gi:83776600]
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4
[SID125299379]
AC50 Counter screen for activity against Aurora B, in dose Measured in Biochemical System Using Scintillation - 2052-06_Inhibitor_Dose_DryPowder_Activity_Set3 [AID588808, Type: confirmatory]aurora kinase B [Homo sapiens] [gi:83776600]
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5
[SID125299379]
AC50 Counter screen for activity against Aurora B, in dose Measured in Biochemical System Using Scintillation - 2052-06_Inhibitor_Dose_DryPowder_Activity_Set3 [AID588808, Type: confirmatory]aurora kinase B [Homo sapiens] [gi:83776600]
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