BRD-K14952051-001-01-7
(CID
53377413
) -
BioAssay Data Summary for Compound
.
BioActivity Outcomes:
Inactive(
1
)
Top Targets:
STKc AGC(
1
)
BioAssay Types:
Confirmatory(
1
)
BioActivity Types:
AC50(
1
)
SAR
Target summary
Data download
Chemical Probe
Active
Inactive
Inconclusive
Unspecified
Total Bioassays: 1 Data Row: 1 Total Pages: 1
#
Substance
Activity
BioAssay
Target
Links
Outcome
Type
Value [μM]
1
[SID
125299427
]
Inactive
AC50
STK-33 Kinase Inhibition Measured in Biochemical System Using Plate Reader - 2052-02_Inhibitor_Dose_DryPowder_Activity_Set3 [AID
602158
, Type: confirmatory]
serine/threonine-protein kinase 33 [Homo sapiens] [gi:
23943882
]
View
X
Row No.
1
Structure
Substance
SID
125299427
CID
53377413
Outcome
Inactive
AC50
[uM]
BioAssay
STK-33 Kinase Inhibition Measured in Biochemical System Using Plate Reader - 2052-02_Inhibitor_Dose_DryPowder_Activity_Set3
AID
602158
BioAssay type
confirmatory
Target
serine/threonine-protein kinase 33 [Homo sapiens] [gi:
23943882
]
PubMed
Data Table
2
[SID
125299427
]
Inactive
AC50
STK-33 Kinase Inhibition Measured in Biochemical System Using Plate Reader - 2052-02_Inhibitor_Dose_DryPowder_Activity_Set3 [AID
602158
, Type: confirmatory]
serine/threonine-protein kinase 33 [Homo sapiens] [gi:
23943882
]
View
X
Row No.
2
Structure
Substance
SID
125299427
CID
53377413
Outcome
Inactive
AC50
[uM]
BioAssay
STK-33 Kinase Inhibition Measured in Biochemical System Using Plate Reader - 2052-02_Inhibitor_Dose_DryPowder_Activity_Set3
AID
602158
BioAssay type
confirmatory
Target
serine/threonine-protein kinase 33 [Homo sapiens] [gi:
23943882
]
PubMed
Data Table
3
[SID
125299427
]
Inactive
AC50
STK-33 Kinase Inhibition Measured in Biochemical System Using Plate Reader - 2052-02_Inhibitor_Dose_DryPowder_Activity_Set3 [AID
602158
, Type: confirmatory]
serine/threonine-protein kinase 33 [Homo sapiens] [gi:
23943882
]
View
X
Row No.
3
Structure
Substance
SID
125299427
CID
53377413
Outcome
Inactive
AC50
[uM]
BioAssay
STK-33 Kinase Inhibition Measured in Biochemical System Using Plate Reader - 2052-02_Inhibitor_Dose_DryPowder_Activity_Set3
AID
602158
BioAssay type
confirmatory
Target
serine/threonine-protein kinase 33 [Homo sapiens] [gi:
23943882
]
PubMed
Data Table