(2-Benzylpiperidin-1-yl)(4-(4-bromophenyl)-1H-1,2,3-triazol-1-yl)methanone (CID 53364489) - BioAssay Data Summary for Compound
.
BioActivity Outcomes:
Active(17)
 
 
Inactive(8)
 
 
Top Targets:
Lipase 3(10)
 
 
 
Lipase(6)
 
 
 
Peptidase S9(2)
 
 
 
luxD(2)
 
 
 
Esterase lipa..(1)
 
 
SAR
Target summary
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 5    Data Row: 25   Total Pages: 1   
Sort: [Click the result table header to sort]
#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID125269114]
 Late stage assay provider results from the probe development effort to identify inhibitors of diacylglycerol lipase, beta (DAGLb): fluorescence-based biochemical gel-based competitive Activity-Based Protein Profiling (ABPP) inhibition of serine hydrolases in mouse brain membrane in vitro set 1 [AID602311, Type: other]Abhd6 gene product [Mus musculus] [gi:31560264]
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2
[SID125269114]
 Late stage assay provider results from the probe development effort to identify inhibitors of diacylglycerol lipase, beta (DAGLb): fluorescence-based biochemical gel-based competitive Activity-Based Protein Profiling (ABPP) inhibition of serine hydrolases in mouse brain membrane in vitro set 1 [AID602311, Type: other]Abhd6 gene product [Mus musculus] [gi:31560264]
View
3
[SID125269114]
 Late stage assay provider results from the probe development effort to identify inhibitors of diacylglycerol lipase, beta (DAGLb): fluorescence-based biochemical gel-based competitive Activity-Based Protein Profiling (ABPP) inhibition of serine hydrolases in mouse brain membrane in vitro set 1 [AID602311, Type: other]Abhd6 gene product [Mus musculus] [gi:31560264]
View
4
[SID125269114]
 Late stage assay provider results from the probe development effort to identify inhibitors of diacylglycerol lipase, beta (DAGLb): fluorescence-based biochemical gel-based competitive Activity-Based Protein Profiling (ABPP) inhibition of serine hydrolases in mouse brain membrane in vitro set 1 [AID602311_1, Type: other]Abhd6 gene product [Mus musculus] [gi:31560264]
View
5
[SID125269114]
 Late stage assay provider results from the probe development effort to identify inhibitors of diacylglycerol lipase, beta (DAGLb): fluorescence-based biochemical gel-based competitive Activity-Based Protein Profiling (ABPP) inhibition of serine hydrolases in mouse brain membrane in vitro set 1 [AID602311_1, Type: other]Abhd6 gene product [Mus musculus] [gi:31560264]
View
6
[SID125269114]
 Late stage assay provider results from the probe development effort to identify inhibitors of diacylglycerol lipase, beta (DAGLb): fluorescence-based biochemical gel-based competitive Activity-Based Protein Profiling (ABPP) inhibition of serine hydrolases in mouse brain membrane in vitro set 1 [AID602311_1, Type: other]Abhd6 gene product [Mus musculus] [gi:31560264]
View
7
[SID125269114]
 Late stage assay provider results from the probe development effort to identify inhibitors of diacylglycerol lipase, beta (DAGLb): fluorescence-based biochemical gel-based competitive Activity-Based Protein Profiling (ABPP) inhibition of serine hydrolases in mouse brain membrane in vitro set 1 [AID602311_3, Type: other]fatty acid amide hydrolase [Mus musculus] [gi:123253900]
View
8
[SID125269114]
 Late stage assay provider results from the probe development effort to identify inhibitors of diacylglycerol lipase, beta (DAGLb): fluorescence-based biochemical gel-based competitive Activity-Based Protein Profiling (ABPP) inhibition of serine hydrolases in mouse brain membrane in vitro set 1 [AID602311_3, Type: other]fatty acid amide hydrolase [Mus musculus] [gi:123253900]
View
9
[SID125269114]
 Late stage assay provider results from the probe development effort to identify inhibitors of diacylglycerol lipase, beta (DAGLb): fluorescence-based biochemical gel-based competitive Activity-Based Protein Profiling (ABPP) inhibition of serine hydrolases in mouse brain membrane in vitro set 1 [AID602311_3, Type: other]fatty acid amide hydrolase [Mus musculus] [gi:123253900]
View
10
[SID125269114]
 Late stage assay provider results from the probe development effort to identify inhibitors of diacylglycerol lipase, beta (DAGLb): fluorescence-based biochemical gel-based competitive Activity-Based Protein Profiling (ABPP) inhibition of DAGLb by enantiomers of KT116 [AID624472_2, Type: other]Abhd6 gene product [Mus musculus] [gi:31560264]
View
11
[SID125269114]
 Late stage assay provider results from the probe development effort to identify inhibitors of diacylglycerol lipase, beta (DAGLb): fluorescence-based biochemical gel-based competitive Activity-Based Protein Profiling (ABPP) inhibition of DAGLb by enantiomers of KT116 [AID624472_2, Type: other]Abhd6 gene product [Mus musculus] [gi:31560264]
View
12
[SID125269114]
 Late stage assay provider results from the probe development effort to identify inhibitors of diacylglycerol lipase, beta (DAGLb): fluorescence-based biochemical gel-based competitive Activity-Based Protein Profiling (ABPP) inhibition of serine hydrolases in mouse brain membrane in vitro set 2 [AID602323, Type: other]Daglb gene product [Mus musculus] [gi:31559956]
View
13
[SID125269114]
 Late stage assay provider results from the probe development effort to identify inhibitors of diacylglycerol lipase, beta (DAGLb): fluorescence-based biochemical gel-based competitive Activity-Based Protein Profiling (ABPP) inhibition of serine hydrolases in mouse brain membrane in vitro set 2 [AID602323, Type: other]Daglb gene product [Mus musculus] [gi:31559956]
View
14
[SID125269114]
 Late stage assay provider results from the probe development effort to identify inhibitors of diacylglycerol lipase, beta (DAGLb): fluorescence-based biochemical gel-based competitive Activity-Based Protein Profiling (ABPP) inhibition of serine hydrolases in mouse brain membrane in vitro set 2 [AID602323_1, Type: other]Daglb gene product [Mus musculus] [gi:31559956]
View
15
[SID125269114]
 Late stage assay provider results from the probe development effort to identify inhibitors of diacylglycerol lipase, beta (DAGLb): fluorescence-based biochemical gel-based competitive Activity-Based Protein Profiling (ABPP) inhibition of serine hydrolases in mouse brain membrane in vitro set 2 [AID602323_1, Type: other]Daglb gene product [Mus musculus] [gi:31559956]
View
16
[SID125269114]
 Late stage assay provider results from the probe development effort to identify inhibitors of diacylglycerol lipase, beta (DAGLb): fluorescence-based biochemical gel-based competitive Activity-Based Protein Profiling (ABPP) inhibition of serine hydrolases in mouse brain membrane in vitro set 2 [AID602323_3, Type: other]Daglb gene product [Mus musculus] [gi:31559956]
View
17
[SID125269114]
 Late stage assay provider results from the probe development effort to identify inhibitors of diacylglycerol lipase, beta (DAGLb): fluorescence-based biochemical gel-based competitive Activity-Based Protein Profiling (ABPP) inhibition of serine hydrolases in mouse brain membrane in vitro set 2 [AID602323_3, Type: other]Daglb gene product [Mus musculus] [gi:31559956]
View
18
[SID125269114]
 Late stage assay provider results from the probe development effort to identify inhibitors of diacylglycerol lipase, beta (DAGLb): fluorescence-based biochemical gel-based competitive Activity-Based Protein Profiling (ABPP) inhibition of DAGLb by enantiomers of KT116 [AID624472, Type: other]Daglb gene product [Mus musculus] [gi:31559956]
View
19
[SID125269114]
 Late stage assay provider results from the probe development effort to identify inhibitors of diacylglycerol lipase, beta (DAGLb): fluorescence-based biochemical gel-based competitive Activity-Based Protein Profiling (ABPP) inhibition of DAGLb by enantiomers of KT116 [AID624472, Type: other]Daglb gene product [Mus musculus] [gi:31559956]
View
20
[SID125269114]
 Late stage assay provider results from the probe development effort to identify inhibitors of diacylglycerol lipase, beta (DAGLb): fluorescence-based biochemical gel-based competitive Activity-Based Protein Profiling (ABPP) inhibition of DAGLb by enantiomers of KT116 [AID624472_1, Type: other]Daglb gene product [Mus musculus] [gi:31559956]
View
21
[SID125269114]
 Late stage assay provider results from the probe development effort to identify inhibitors of diacylglycerol lipase, beta (DAGLb): fluorescence-based biochemical gel-based competitive Activity-Based Protein Profiling (ABPP) inhibition of DAGLb by enantiomers of KT116 [AID624472_1, Type: other]Daglb gene product [Mus musculus] [gi:31559956]
View
22
[SID125269114]
 Late stage assay provider results from the probe development effort to identify inhibitors of diacylglycerol lipase, beta (DAGLb): fluorescence-based biochemical gel-based competitive Activity-Based Protein Profiling (ABPP) inhibition of serine hydrolases in mouse brain membrane in vitro set 1 [AID602311_6, Type: other]monoacylglycerol lipase ABHD12 [Mus musculus] [gi:159110817]
View
23
[SID125269114]
 Late stage assay provider results from the probe development effort to identify inhibitors of diacylglycerol lipase, beta (DAGLb): fluorescence-based biochemical gel-based competitive Activity-Based Protein Profiling (ABPP) inhibition of serine hydrolases in mouse brain membrane in vitro set 1 [AID602311_6, Type: other]monoacylglycerol lipase ABHD12 [Mus musculus] [gi:159110817]
View
24
[SID125269114]
 Late stage assay provider results from the probe development effort to identify inhibitors of diacylglycerol lipase, beta (DAGLb): fluorescence-based biochemical gel-based competitive Activity-Based Protein Profiling (ABPP) inhibition of serine hydrolases in mouse brain membrane in vitro set 1 [AID602311_6, Type: other]monoacylglycerol lipase ABHD12 [Mus musculus] [gi:159110817]
View
25
[SID125269114]
 Late stage assay provider results from the probe development effort to identify inhibitors of diacylglycerol lipase, beta (DAGLb): fluorescence-based biochemical gel-based competitive Activity-Based Protein Profiling (ABPP) inhibition of recombinant anti-target ABHD11 in vitro set 1 [AID602301, Type: other]Abhydrolase domain containing 11 [Mus musculus] [gi:47682716]
View
26
[SID125269114]
 Late stage assay provider results from the probe development effort to identify inhibitors of diacylglycerol lipase, beta (DAGLb): fluorescence-based biochemical gel-based competitive Activity-Based Protein Profiling (ABPP) inhibition of recombinant anti-target ABHD11 in vitro set 1 [AID602301, Type: other]Abhydrolase domain containing 11 [Mus musculus] [gi:47682716]
View
27
[SID125269114]
 Late stage assay provider results from the probe development effort to identify inhibitors of diacylglycerol lipase, beta (DAGLb): fluorescence-based biochemical gel-based competitive Activity-Based Protein Profiling (ABPP) inhibition of serine hydrolases in mouse brain membrane in vitro set 2 [AID602323_2, Type: other]Abhd6 gene product [Mus musculus] [gi:31560264]
View
28
[SID125269114]
 Late stage assay provider results from the probe development effort to identify inhibitors of diacylglycerol lipase, beta (DAGLb): fluorescence-based biochemical gel-based competitive Activity-Based Protein Profiling (ABPP) inhibition of serine hydrolases in mouse brain membrane in vitro set 2 [AID602323_2, Type: other]Abhd6 gene product [Mus musculus] [gi:31560264]
View
29
[SID125269114]
 Late stage assay provider results from the probe development effort to identify inhibitors of diacylglycerol lipase, beta (DAGLb): fluorescence-based biochemical gel-based competitive Activity-Based Protein Profiling (ABPP) inhibition of serine hydrolases in mouse brain membrane in vitro set 2 [AID602323_4, Type: other]platelet-activating factor acetylhydrolase precursor [Mus musculus] [gi:31980752]
View
30
[SID125269114]
 Late stage assay provider results from the probe development effort to identify inhibitors of diacylglycerol lipase, beta (DAGLb): fluorescence-based biochemical gel-based competitive Activity-Based Protein Profiling (ABPP) inhibition of serine hydrolases in mouse brain membrane in vitro set 2 [AID602323_4, Type: other]platelet-activating factor acetylhydrolase precursor [Mus musculus] [gi:31980752]
View
31
[SID136946704]
 Late stage assay provider results from the probe development effort to identify inhibitors of diacylglycerol lipase, beta (DAGLb): fluorescence-based biochemical gel-based competitive Activity-Based Protein Profiling (ABPP) inhibition of DAGLb by enantiomers of KT116 [AID624472, Type: other]Daglb gene product [Mus musculus] [gi:31559956]
View
32
[SID136946704]
 Late stage assay provider results from the probe development effort to identify inhibitors of diacylglycerol lipase, beta (DAGLb): fluorescence-based biochemical gel-based competitive Activity-Based Protein Profiling (ABPP) inhibition of DAGLb by enantiomers of KT116 [AID624472, Type: other]Daglb gene product [Mus musculus] [gi:31559956]
View
33
[SID136946704]
 Late stage assay provider results from the probe development effort to identify inhibitors of diacylglycerol lipase, beta (DAGLb): fluorescence-based biochemical gel-based competitive Activity-Based Protein Profiling (ABPP) inhibition of DAGLb by enantiomers of KT116 [AID624472_1, Type: other]Daglb gene product [Mus musculus] [gi:31559956]
View
34
[SID136946704]
 Late stage assay provider results from the probe development effort to identify inhibitors of diacylglycerol lipase, beta (DAGLb): fluorescence-based biochemical gel-based competitive Activity-Based Protein Profiling (ABPP) inhibition of DAGLb by enantiomers of KT116 [AID624472_1, Type: other]Daglb gene product [Mus musculus] [gi:31559956]
View
35
[SID125269114]
 Late stage assay provider results from the probe development effort to identify inhibitors of diacylglycerol lipase, beta (DAGLb): fluorescence-based biochemical gel-based competitive Activity-Based Protein Profiling (ABPP) inhibition of overexpressed DAGLb in vitro set 1 [AID602302, Type: other]Daglb gene product [Mus musculus] [gi:31559956]
View
36
[SID125269114]
 Late stage assay provider results from the probe development effort to identify inhibitors of diacylglycerol lipase, beta (DAGLb): fluorescence-based biochemical gel-based competitive Activity-Based Protein Profiling (ABPP) inhibition of overexpressed DAGLb in vitro set 1 [AID602302, Type: other]Daglb gene product [Mus musculus] [gi:31559956]
View
37
[SID136946704]
 Late stage assay provider results from the probe development effort to identify inhibitors of diacylglycerol lipase, beta (DAGLb): fluorescence-based biochemical gel-based competitive Activity-Based Protein Profiling (ABPP) inhibition of DAGLb by enantiomers of KT116 [AID624472_2, Type: other]Abhd6 gene product [Mus musculus] [gi:31560264]
View
38
[SID136946704]
 Late stage assay provider results from the probe development effort to identify inhibitors of diacylglycerol lipase, beta (DAGLb): fluorescence-based biochemical gel-based competitive Activity-Based Protein Profiling (ABPP) inhibition of DAGLb by enantiomers of KT116 [AID624472_2, Type: other]Abhd6 gene product [Mus musculus] [gi:31560264]
View
39
[SID136946703]
 Late stage assay provider results from the probe development effort to identify inhibitors of diacylglycerol lipase, beta (DAGLb): fluorescence-based biochemical gel-based competitive Activity-Based Protein Profiling (ABPP) inhibition of DAGLb by enantiomers of KT116 [AID624472_2, Type: other]Abhd6 gene product [Mus musculus] [gi:31560264]
View
40
[SID136946703]
 Late stage assay provider results from the probe development effort to identify inhibitors of diacylglycerol lipase, beta (DAGLb): fluorescence-based biochemical gel-based competitive Activity-Based Protein Profiling (ABPP) inhibition of DAGLb by enantiomers of KT116 [AID624472_2, Type: other]Abhd6 gene product [Mus musculus] [gi:31560264]
View
41
[SID136946703]
 Late stage assay provider results from the probe development effort to identify inhibitors of diacylglycerol lipase, beta (DAGLb): fluorescence-based biochemical gel-based competitive Activity-Based Protein Profiling (ABPP) inhibition of DAGLb by enantiomers of KT116 [AID624472, Type: other]Daglb gene product [Mus musculus] [gi:31559956]
View
42
[SID136946703]
 Late stage assay provider results from the probe development effort to identify inhibitors of diacylglycerol lipase, beta (DAGLb): fluorescence-based biochemical gel-based competitive Activity-Based Protein Profiling (ABPP) inhibition of DAGLb by enantiomers of KT116 [AID624472, Type: other]Daglb gene product [Mus musculus] [gi:31559956]
View
43
[SID136946703]
 Late stage assay provider results from the probe development effort to identify inhibitors of diacylglycerol lipase, beta (DAGLb): fluorescence-based biochemical gel-based competitive Activity-Based Protein Profiling (ABPP) inhibition of DAGLb by enantiomers of KT116 [AID624472_1, Type: other]Daglb gene product [Mus musculus] [gi:31559956]
View
44
[SID136946703]
 Late stage assay provider results from the probe development effort to identify inhibitors of diacylglycerol lipase, beta (DAGLb): fluorescence-based biochemical gel-based competitive Activity-Based Protein Profiling (ABPP) inhibition of DAGLb by enantiomers of KT116 [AID624472_1, Type: other]Daglb gene product [Mus musculus] [gi:31559956]
View
45
[SID125269114]
 Late stage assay provider results from the probe development effort to identify inhibitors of diacylglycerol lipase, beta (DAGLb): fluorescence-based biochemical gel-based competitive Activity-Based Protein Profiling (ABPP) inhibition of serine hydrolases in mouse brain membrane in vitro set 1 [AID602311_5, Type: other]monoacylglycerol lipase ABHD12 [Mus musculus] [gi:159110817]
View
46
[SID125269114]
 Late stage assay provider results from the probe development effort to identify inhibitors of diacylglycerol lipase, beta (DAGLb): fluorescence-based biochemical gel-based competitive Activity-Based Protein Profiling (ABPP) inhibition of serine hydrolases in mouse brain membrane in vitro set 1 [AID602311_5, Type: other]monoacylglycerol lipase ABHD12 [Mus musculus] [gi:159110817]
View
47
[SID125269114]
 Late stage assay provider results from the probe development effort to identify inhibitors of diacylglycerol lipase, beta (DAGLb): fluorescence-based biochemical gel-based competitive Activity-Based Protein Profiling (ABPP) inhibition of serine hydrolases in mouse brain membrane in vitro set 1 [AID602311_5, Type: other]monoacylglycerol lipase ABHD12 [Mus musculus] [gi:159110817]
View
48
[SID125269114]
 Late stage assay provider results from the probe development effort to identify inhibitors of diacylglycerol lipase, beta (DAGLb): fluorescence-based biochemical gel-based competitive Activity-Based Protein Profiling (ABPP) inhibition of serine hydrolases in mouse brain membrane in vitro set 1 [AID602311_8, Type: other]acyl-protein thioesterase 1 [Mus musculus] [gi:6678760]
View
49
[SID125269114]
 Late stage assay provider results from the probe development effort to identify inhibitors of diacylglycerol lipase, beta (DAGLb): fluorescence-based biochemical gel-based competitive Activity-Based Protein Profiling (ABPP) inhibition of serine hydrolases in mouse brain membrane in vitro set 1 [AID602311_8, Type: other]acyl-protein thioesterase 1 [Mus musculus] [gi:6678760]
View
50
[SID125269114]
 Late stage assay provider results from the probe development effort to identify inhibitors of diacylglycerol lipase, beta (DAGLb): fluorescence-based biochemical gel-based competitive Activity-Based Protein Profiling (ABPP) inhibition of serine hydrolases in mouse brain membrane in vitro set 1 [AID602311_8, Type: other]acyl-protein thioesterase 1 [Mus musculus] [gi:6678760]
View