BRD-K22549930-001-01-8 (CID 53348007) - BioAssay Data Summary for Compound
.
BioActivity Outcomes:
Active(2)
 
 
Inactive(1)
 
 
Top Targets:
STKc AGC(2)
 
 
 
STKc PKA(1)
 
 
BioAssay Types:
Confirmatory(3)
 
 
 
BioActivity Types:
AC50(3)
 
 
 
SAR
Target summary
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 3    Data Row: 3   Total Pages: 1   
Sort: [Click the result table header to sort]
#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID125081984]
AC50 6.73Protein Kinase A Activity Assay Measured in Biochemical System Using Plate Reader - 2052-04_Inhibitor_Dose_DryPowder_Activity_Set2 [AID588629, Type: confirmatory]cAMP-dependent protein kinase catalytic subunit alpha isoform 1 [Homo sapiens] [gi:4506055]
View
2
[SID125081984]
AC50 6.73Protein Kinase A Activity Assay Measured in Biochemical System Using Plate Reader - 2052-04_Inhibitor_Dose_DryPowder_Activity_Set2 [AID588629, Type: confirmatory]cAMP-dependent protein kinase catalytic subunit alpha isoform 1 [Homo sapiens] [gi:4506055]
View
3
[SID125081984]
AC50 8.51STK-33 Kinase Inhibition Measured in Biochemical System Using Plate Reader - 2052-02_Inhibitor_Dose_DryPowder_Activity_Set2 [AID588480, Type: confirmatory]serine/threonine-protein kinase 33 [Homo sapiens] [gi:23943882]
View
4
[SID125081984]
AC50 8.51STK-33 Kinase Inhibition Measured in Biochemical System Using Plate Reader - 2052-02_Inhibitor_Dose_DryPowder_Activity_Set2 [AID588480, Type: confirmatory]serine/threonine-protein kinase 33 [Homo sapiens] [gi:23943882]
View
5
[SID125081984]
AC50 8.51STK-33 Kinase Inhibition Measured in Biochemical System Using Plate Reader - 2052-02_Inhibitor_Dose_DryPowder_Activity_Set2 [AID588480, Type: confirmatory]serine/threonine-protein kinase 33 [Homo sapiens] [gi:23943882]
View
6
[SID125299440]
AC50 STK-33 Kinase Inhibition Measured in Biochemical System Using Plate Reader - 2052-02_Inhibitor_Dose_DryPowder_Activity_Set3 [AID602158, Type: confirmatory]serine/threonine-protein kinase 33 [Homo sapiens] [gi:23943882]
View
7
[SID125299440]
AC50 STK-33 Kinase Inhibition Measured in Biochemical System Using Plate Reader - 2052-02_Inhibitor_Dose_DryPowder_Activity_Set3 [AID602158, Type: confirmatory]serine/threonine-protein kinase 33 [Homo sapiens] [gi:23943882]
View
8
[SID125299440]
AC50 STK-33 Kinase Inhibition Measured in Biochemical System Using Plate Reader - 2052-02_Inhibitor_Dose_DryPowder_Activity_Set3 [AID602158, Type: confirmatory]serine/threonine-protein kinase 33 [Homo sapiens] [gi:23943882]
View