CHEMBL1771112 (CID 53327908) - BioAssay Data Summary for Compound
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BioActivity Outcomes:
Active(8)
 
 
Top Targets:
7TM GPCR Srx(3)
 
 
7TM GPCR Srsx(1)
 
 
BioAssay Types:
Literature(8)
 
 
BioActivity Types:
Ki(8)
 
 
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Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 8    Data Row: 8   Total Pages: 1   
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#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID131281795]
Ki 0.00012Displacement of [3H]Spiperone from human dopamine D3 receptor expressed in CHO cells [AID594007, Type: Literature]D(3) dopamine receptor [gi:1169206]
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2
[SID131281795]
Ki 0.00012Displacement of [3H]Spiperone from human dopamine D3 receptor expressed in CHO cells [AID594007, Type: Literature]D(3) dopamine receptor [gi:1169206]
View
3
[SID131281795]
Ki 0.00012Displacement of [3H]Spiperone from human dopamine D3 receptor expressed in CHO cells [AID594007, Type: Literature]D(3) dopamine receptor [gi:1169206]
View
4
[SID131281795]
Ki 0.00012Displacement of [3H]Spiperone from human dopamine D3 receptor expressed in CHO cells [AID594007, Type: Literature]D(3) dopamine receptor [gi:1169206]
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5
[SID131281795]
Ki 0.0022Displacement of [3H]Prazosin from pig adrenergic alpha1 receptor [AID594011, Type: Literature]
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6
[SID131281795]
Ki 0.0034Displacement of [3H]Spiperone from human dopamine D4.4 receptor expressed in CHO cells [AID594008, Type: Literature]
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7
[SID131281795]
Ki 0.0071Displacement of [3H]Spiperone from human dopamine D2 long receptor expressed in CHO cells [AID594005, Type: Literature]D(2) dopamine receptor [gi:118206]
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8
[SID131281795]
Ki 0.0071Displacement of [3H]Spiperone from human dopamine D2 long receptor expressed in CHO cells [AID594005, Type: Literature]D(2) dopamine receptor [gi:118206]
View
9
[SID131281795]
Ki 0.0071Displacement of [3H]Spiperone from human dopamine D2 long receptor expressed in CHO cells [AID594005, Type: Literature]D(2) dopamine receptor [gi:118206]
View
10
[SID131281795]
Ki 0.0071Displacement of [3H]Spiperone from human dopamine D2 long receptor expressed in CHO cells [AID594005, Type: Literature]D(2) dopamine receptor [gi:118206]
View
11
[SID131281795]
Ki 0.0071Displacement of [3H]Spiperone from human dopamine D2 long receptor expressed in CHO cells [AID594005, Type: Literature]D(2) dopamine receptor [gi:118206]
View
12
[SID131281795]
Ki 0.013Displacement of [3H]Spiperone from human dopamine D2 short receptor expressed in CHO cells [AID594006, Type: Literature]D(2) dopamine receptor [gi:118206]
View
13
[SID131281795]
Ki 0.013Displacement of [3H]Spiperone from human dopamine D2 short receptor expressed in CHO cells [AID594006, Type: Literature]D(2) dopamine receptor [gi:118206]
View
14
[SID131281795]
Ki 0.013Displacement of [3H]Spiperone from human dopamine D2 short receptor expressed in CHO cells [AID594006, Type: Literature]D(2) dopamine receptor [gi:118206]
View
15
[SID131281795]
Ki 0.013Displacement of [3H]Spiperone from human dopamine D2 short receptor expressed in CHO cells [AID594006, Type: Literature]D(2) dopamine receptor [gi:118206]
View
16
[SID131281795]
Ki 0.013Displacement of [3H]Spiperone from human dopamine D2 short receptor expressed in CHO cells [AID594006, Type: Literature]D(2) dopamine receptor [gi:118206]
View
17
[SID131281795]
Ki 0.013Displacement of [3H]WAY-100635 from pig 5-HT1A receptor [AID594009, Type: Literature]
View
18
[SID131281795]
Ki 0.16Displacement of [3H]Ketanserin from pig 5-HT2 receptor [AID594010, Type: Literature]5-hydroxytryptamine receptor 2A [gi:1703009]
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19
[SID131281795]
Ki 0.38Displacement of [3H]SCH-23390 from dopamine D1 receptor in pig striatal membranes [AID594004, Type: Literature]D(1A) dopamine receptor [gi:1706296]
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