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AGN-PC-09Q7SF (CID 53304409) - Compound BioActivity Data
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BioActivity Outcomes:
Active(2)
 
 
Unspecified(2)
 
 
Top Targets:
Esterase lipa..(2)
 
 
BioAssay Types:
Literature(4)
 
 
 
BioActivity Types:
IC50(2)
 
 
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 4    Data Row: 4   Total Pages: 1   
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#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID131274657]
IC50 0.0244Inhibition of equine serum BuChE assessed as inhibition of butyrylthiocholine chloride substrate hydrolysis incubated for 15 mins before substrate addition measured by spectrophotometry [AID601100, Type: Literature]Cholinesterase [gi:21362409]
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2
[SID131274657]
IC50 0.1044Inhibition of electric eel AChE assessed as inhibition of acetylthiocholine chloride substrate hydrolysis incubated for 15 mins before substrate addition measured by spectrophotometry [AID601099, Type: Literature]Acetylcholinesterase [gi:14916521]
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3
[SID131274657]
Selectivity index, ratio of IC50 for electric eel AChE to IC50 for equine serum BuChE [AID601101, Type: Literature]
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4
[SID131274657]
Antioxidant activity against AAPH-induced peroxyl radical assessed as trolox equivalent at 1 to 5 uM after 15 mins by oxygen radical absorbance capacity-fluorescein assay [AID601104, Type: Literature]
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