Bookmark and Share
CHEBI:51074 (CID 53278) - Compound BioActivity Data
.
BioActivity Outcomes:
Active(7)
 
 
Inactive(212)
 
 
Inconclusive(25)
 
 
Unspecified(4)
 
 
Top Targets:
p450(17)
 
 
 
HSD10-like SD..(10)
 
 
Git3(6)
 
 
 
ampC(6)
 
 
NR LBD GR(6)
 
 
BioAssay Types:
Confirmatory(217)
 
 
 
 
 
Screening(2)
 
 
Literature(2)
 
 
BioActivity Types:
Potency(149)
 
 
 
 
 
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 108    Data Row: 248   Total Pages: 5   Display: Page     
Sort: [Click the result table header to sort]
#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID124882771]
Potency 0.0596qHTS for Inhibitors of human tyrosyl-DNA phosphodiesterase 1 (TDP1): qHTS in cells in absence of CPT [AID686978, Type: confirmatory]TDP1 protein [Homo sapiens] [gi:79154014]
View
2
[SID124882771]
Potency 0.0944qHTS for Inhibitors of human tyrosyl-DNA phosphodiesterase 1 (TDP1): qHTS in cells in presence of CPT [AID686979, Type: confirmatory]TDP1 protein [Homo sapiens] [gi:79154014]
View
3
[SID11113078]
Cell signaling CRE-BLA (Fsk stim) [AID662, Type: confirmatory]
View
4
[SID11113078]
qHTS Assay for Spectroscopic Profiling in 4-MU Spectral Region [AID589, Type: other]
View
5
[SID11113078]
qHTS Assay for Spectroscopic Profiling in A350 Spectral Region [AID590, Type: other]
View
6
[SID11112178]
Cell signaling CRE-BLA (Fsk stim) [AID662, Type: confirmatory]
View
7
[SID11111007]
Cell signaling CRE-BLA (Fsk stim) [AID662, Type: confirmatory]
View
8
[SID11111007]
Potency 0.1259qHTS Assay for Agonists of the Thyroid Stimulating Hormone Receptor [AID926, Type: confirmatory]thyroid stimulating hormone receptor [Homo sapiens] [gi:38016895]
View
9
[SID11112178]
Cytochrome panel assay with activity outcomes [AID1851, Type: other]
View
10
[SID103296084]
Toxicity found after a single im injection. The total number of deaths were counted after 7 days and LD50 was determined by probit analysis; 82.9-163.4 [AID123251, Type: Literature]
View
11
[SID103296084]
Inhibition of [3H]colchicine binding to microtubule protein tubulin [AID214375, Type: Literature]
View
12
[SID11112178]
Potency qHTS for Inhibitors of binding or entry into cells for Lassa Virus [AID720533, Type: confirmatory]
View
13
[SID124882771]
Potency qHTS for Inhibitors of binding or entry into cells for Lassa Virus [AID720533, Type: confirmatory]
View
14
[SID26754264]
Potency qHTS Assay for Allosteric/Competitive Inhibitors of Caspase-1: Spectroscopic Profiling in AFC Spectral Region [AID923, Type: confirmatory]
View
15
[SID26754264]
Potency Counterscreen qHTS for Inhibitors of Tau Fibril Formation, Fluorescence Polarization [AID1463, Type: confirmatory]
View
16
[SID26754264]
Potency qHTS Assay for Compounds Blocking the Interaction Between CBF-beta and RUNX1 for the Treatment of Acute Myeloid Leukemia [AID1477, Type: confirmatory]
View
17
[SID11113078]
qHTS Assay for Spectroscopic Profiling in Texas Red Spectral Region [AID587, Type: other]
View
18
[SID11113078]
qHTS Assay for Spectroscopic Profiling in Resorufin Spectral Region [AID588, Type: other]
View
19
[SID11111007]
Ubiquitin-GFP Assay [AID526, Type: confirmatory]
View
20
[SID11111007]
qHTS Assay for Spectroscopic Profiling in Texas Red Spectral Region [AID587, Type: other]
View
21
[SID26754264]
Potency Quantitative High-Throughput Screen for Regulators of Epigenetic Control [AID1865, Type: confirmatory]
View
22
[SID26754264]
Potency qHTS Assay for Compounds that Induce Erasure of Genomic Imprints [AID1948, Type: confirmatory]
View
23
[SID11113078]
qHTS Assay for Spectroscopic Profiling in Fluorescein Spectral Region [AID593, Type: other]
View
24
[SID11113078]
qHTS Assay for Spectroscopic Profiling in Rhodamine Spectral Region [AID594, Type: confirmatory]
View
25
[SID11113078]
qHTS Assay for Disrupters of an Hsp90 Co-Chaperone Interaction [AID595, Type: confirmatory]
View
26
[SID11113078]
qHTS Assay for Epigenetic Modulators [AID597, Type: confirmatory]
View
27
[SID11113078]
qHTS Assay for Inhibitors of DNA Polymerase III Holoenzyme System [AID603, Type: confirmatory]
View
28
[SID11112178]
Potency Quantitative High-Throughput Screen for Regulators of Epigenetic Control [AID1865, Type: confirmatory]
View
29
[SID11112178]
Potency qHTS Assay for Compounds that Induce Erasure of Genomic Imprints [AID1948, Type: confirmatory]
View
30
[SID11113078]
qHTS Assay for Spectroscopic Profiling in A488 Spectral Region [AID591, Type: other]
View
31
[SID11113078]
qHTS Assay for Spectroscopic Profiling in A647 Spectral Region [AID592, Type: other]
View
32
[SID11112178]
Potency qHTS Assay for Lipid Storage Modulators [AID1519, Type: confirmatory]
View
33
[SID11112178]
Potency qHTS Assay for Allosteric/Competitive Inhibitors of Caspase-1: Spectroscopic Profiling in AFC Spectral Region [AID923, Type: confirmatory]
View
34
[SID11112178]
Potency qHTS Assay for Compounds Blocking the Interaction Between CBF-beta and RUNX1 for the Treatment of Acute Myeloid Leukemia [AID1477, Type: confirmatory]
View
35
[SID11112178]
qHTS Assay for Spectroscopic Profiling in 4-MU Spectral Region [AID589, Type: other]
View
36
[SID11112178]
qHTS Assay for Spectroscopic Profiling in A350 Spectral Region [AID590, Type: other]
View
37
[SID11112178]
qHTS Assay for Spectroscopic Profiling in A488 Spectral Region [AID591, Type: other]
View
38
[SID11112178]
qHTS Assay for Spectroscopic Profiling in A647 Spectral Region [AID592, Type: other]
View
39
[SID11112178]
Potency qHTS Assay for Enhancers of SMN2 Splice Variant Expression [AID1458, Type: confirmatory]survival motor neuron protein isoform d [Homo sapiens] [gi:10937869]
View
40
[SID11112178]
Potency qHTS Assay for Inhibitors of Bacillus subtilis Sfp phosphopantetheinyl transferase (PPTase) [AID1490, Type: confirmatory]phosphopantetheinyl transferase [Bacillus subtilis] [gi:10954339]
View
41
[SID26754264]
Potency qHTS Assay for Inhibitors of Bacillus subtilis Sfp phosphopantetheinyl transferase (PPTase) [AID1490, Type: confirmatory]phosphopantetheinyl transferase [Bacillus subtilis] [gi:10954339]
View
42
[SID124882771]
Potency qHTS for inhibitors of Vif-A3G interactions: Validation [AID588379, Type: confirmatory]DNA dC->dU-editing enzyme APOBEC-3G [Homo sapiens] [gi:13399304]
View
43
[SID11112178]
Potency qHTS Assay for Inhibitors and Substrates of Cytochrome P450 3A4 [AID884, Type: confirmatory]cytochrome P450 3A4 isoform 1 [Homo sapiens] [gi:13435386]
View
44
[SID11112178]
Potency qHTS Assay for Activators of Cytochrome P450 3A4 [AID885, Type: confirmatory]cytochrome P450 3A4 isoform 1 [Homo sapiens] [gi:13435386]
View
45
[SID11112178]
Cytochrome panel assay with activity outcomes [AID1851_3, Type: other]cytochrome P450 3A4 isoform 1 [Homo sapiens] [gi:13435386]
View
46
[SID26754264]
Potency qHTS Assay for Inhibitors and Substrates of Cytochrome P450 3A4 [AID884, Type: confirmatory]cytochrome P450 3A4 isoform 1 [Homo sapiens] [gi:13435386]
View
47
[SID26754264]
Potency qHTS Assay for Activators of Cytochrome P450 3A4 [AID885, Type: confirmatory]cytochrome P450 3A4 isoform 1 [Homo sapiens] [gi:13435386]
View
48
[SID11112178]
Potency qHTS Assay for Inhibitors and Substrates of Cytochrome P450 2C9 [AID883, Type: confirmatory]cytochrome P450 2C9 precursor [Homo sapiens] [gi:13699818]
View
49
[SID11112178]
Cytochrome panel assay with activity outcomes [AID1851_5, Type: other]cytochrome P450 2C9 precursor [Homo sapiens] [gi:13699818]
View
50
[SID11113078]
Potency qHTS Assay for Inhibitors and Substrates of Cytochrome P450 2C9 [AID883, Type: confirmatory]cytochrome P450 2C9 precursor [Homo sapiens] [gi:13699818]
View