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CHEMBL2431120 (CID 53245590) - Compound BioActivity Data
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BioActivity Outcomes:
Probe(1)
 
 
Active(3)
 
 
Inactive(3)
 
 
Top Targets:
7TM GPCR Srv(5)
 
 
 
 
BioAssay Types:
Confirmatory(6)
 
 
 
Summary(1)
 
 
BioActivity Types:
EC50(5)
 
 
 
IC50(1)
 
 
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 5    Data Row: 7   Total Pages: 1   
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#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID134225039]
Summary Assay for Selective Agonists of NTR1 [AID493055, Type: summary]neurotensin receptor type 1 [Homo sapiens] [gi:110611243]
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2
[SID134225039]
EC50_Mean 1.89SAR analysis of small molecule Agonists NTR1 in a image based assay set 3 [AID602356, Type: confirmatory]neurotensin receptor type 1 [Homo sapiens] [gi:110611243]
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3
[SID124360477]
EC50_Mean 2.18SAR analysis of small molecule Agonists NTR1 in a image based assay set 3 [AID602356, Type: confirmatory]neurotensin receptor type 1 [Homo sapiens] [gi:110611243]
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4
[SID124360477]
EC50_Mean 3.8SAR analysis of small molecule agonists of the NTR1 receptor via a luminescent beta-arrestin assay [AID602427, Type: confirmatory]neurotensin receptor type 1 [Homo sapiens] [gi:110611243]
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5
[SID134225039]
IC50_Mean 25.4SAR analysis of small molecule agonists of the NTR1 receptor via a luminescent cytotoxicity assay [AID602482, Type: confirmatory]neurotensin receptor type 1 [Homo sapiens] [gi:110611243]
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6
[SID124360477]
EC50_Mean 80SAR analysis of small molecule NTR1 agonists in a image based NTR2 selectivity assay set 2 [AID602334, Type: confirmatory]neurotensin receptor type 2 [Homo sapiens] [gi:6912538]
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7
[SID134225039]
EC50_Mean 80SAR analysis of small molecule NTR1 agonists in a image based NTR2 selectivity assay set 2 [AID602334, Type: confirmatory]neurotensin receptor type 2 [Homo sapiens] [gi:6912538]
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