Bookmark and Share
Proscillaridin (CID 5284613) - Compound BioActivity Data
.
BioActivity Outcomes:
Active(29)
 
 
Inactive(35)
 
 
Inconclusive(35)
 
 
Unspecified(146)
 
 
Top Targets:
7TM GPCR Srsx(17)
 
 
 
7TM GPCR Srx(16)
 
 
p450(10)
 
 
 
 
NR LBD ER(9)
 
 
 
 
NR LBD PPAR(8)
 
 
BioAssay Types:
Confirmatory(184)
 
 
 
 
 
Summary(24)
 
 
 
 
Literature(18)
 
 
 
Screening(2)
 
 
BioActivity Types:
IC50(119)
 
 
 
Potency(86)
 
 
 
 
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 245    Data Row: 245   Total Pages: 13   Display: Page     
Sort: [Click the result table header to sort]
#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID144203993]
Potency-Replicate_1 0.0057qHTS assay to identify small molecule antagonists of the androgen receptor (AR) signaling pathway - cell viability counter screen [AID743033, Type: confirmatory]
View
2
[SID170465956]
Potency-Replicate_1 0.006qHTS assay for small molecule activators of the heat shock response signaling pathway - cell viability counter screen [AID743209, Type: confirmatory]
View
3
[SID144203993]
Potency-Replicate_1 0.0072qHTS assay for small molecule agonists of the p53 signaling pathway - cell viability [AID651633, Type: confirmatory]
View
4
[SID170465956]
Potency-Replicate_1 0.0106qHTS assay to identify small molecule antagonists of the farnesoid-X-receptor (FXR) signaling pathway - cell viability counter screen [AID743221, Type: confirmatory]
View
5
[SID170465956]
Potency-Replicate_1 0.0119qHTS assay to identify small molecule antagonists of the peroxisome proliferator-activated receptor delta (PPARd) signaling pathway - cell viability counter screen [AID743213, Type: confirmatory]
View
6
[SID170465956]
Potency-Replicate_1 0.0119qHTS assay to identify small molecule antagonists of the peroxisome proliferator-activated receptor gamma (PPARg) signaling pathway - cell viability counter screen [AID743194, Type: confirmatory]
View
7
[SID170465956]
Potency-Replicate_1 0.0133qHTS assay to identify small molecule agonists of the vitamin D receptor (VDR) signaling pathway - cell viability counter screen [AID743224, Type: confirmatory]
View
8
[SID170465956]
Potency-Replicate_1 0.0134qHTS assay to identify small molecule antagonists of the vitamin D receptor (VDR) signaling pathway - cell viability counter screen [AID743225, Type: confirmatory]
View
9
[SID170465956]
Potency-Replicate_1 0.0188qHTS assay to identify small molecule agonists of the peroxisome proliferator-activated receptor delta (PPARd) signaling pathway - cell viability counter screen [AID743211, Type: confirmatory]
View
10
[SID170465956]
Potency-Replicate_1 0.0211qHTS assay for small molecule agonists of the antioxidant response element (ARE) signaling pathway - cell viability counter screen [AID743203, Type: confirmatory]
View
11
[SID144203993]
Potency-Replicate_1 0.0227qHTS assay for small molecules that induce genotoxicity in human embryonic kidney cells expressing luciferase-tagged ATAD5 - cell viability [AID651634, Type: confirmatory]
View
12
[SID144203993]
Potency-Replicate_1 0.0574qHTS assay to identify small molecule antagonists of the glucocorticoid receptor (GR) signaling pathway [AID720692, Type: confirmatory]glucocorticoid receptor [Homo sapiens] [gi:311348376]
View
13
[SID103558584]
IC50 0.06Cytotoxicity against human HCT116 cells after 72 hrs by FMCA method [AID471512, Type: Literature]
View
14
[SID144203993]
Potency-Replicate_1 0.0639qHTS assay for small molecule disruptors of the mitochondrial membrane potential [AID720635, Type: confirmatory]
View
15
[SID144203993]
Ratio Potency (uM) 0.0868291qHTS assay for small molecule disruptors of the mitochondrial membrane potential: Summary [AID720637, Type: summary]
View
16
[SID103558584]
IC50 0.088DRUGMATRIX: ATPase, Na+/K+ enzyme inhibition (substrate: ATP) [AID625210, Type: confirmatory]
View
17
[SID144203993]
Potency-Replicate_1 0.091qHTS assay to identify small molecule antagonists of the glucocorticoid receptor (GR) signaling pathway - cell viability counter screen [AID720693, Type: confirmatory]
View
18
[SID144203993]
Potency-Replicate_1 0.1012qHTS assay for identifying genotoxic compounds that show differential cytotoxicity against isogenic chicken DT40 cell lines with known DNA damage response pathways - Rev3 mutant cell line [AID743014, Type: confirmatory]
View
19
[SID144203993]
Potency-Replicate_1 0.1274qHTS assay for identifying genotoxic compounds that show differential cytotoxicity against isogenic chicken DT40 cell lines with known DNA damage response pathways - Rad54/Ku70 mutant cell line [AID743015, Type: confirmatory]
View
20
[SID144203993]
Potency-Replicate_1 0.1274qHTS assay for identifying genotoxic compounds that show differential cytotoxicity against isogenic chicken DT40 cell lines with known DNA damage response pathways - wild type cell line [AID743012, Type: confirmatory]
View