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N-arachidonylglycine (CID 5283389) - Compound BioActivity Data
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BioActivity Outcomes:
Active(33)
 
 
Inactive(435)
 
 
Inconclusive(82)
 
 
Unspecified(20)
 
 
Top Targets:
p450(11)
 
 
 
NR LBD TR(11)
 
 
PLN02808(10)
 
 
Tubulin-bindi..(9)
 
 
 
HELICc(9)
 
 
 
BioAssay Types:
Confirmatory(395)
 
 
 
 
 
Literature(97)
 
 
 
 
 
Screening(35)
 
 
Summary(25)
 
 
 
BioActivity Types:
Potency(381)
 
 
 
 
 
IC50(7)
 
 
Ki(1)
 
 
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 373    Data Row: 570   Total Pages: 12   Display: Page     
Sort: [Click the result table header to sort]
#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID50105803]
Potency 0.5012qHTS for Inhibitors of Polymerase Eta [AID588591, Type: confirmatory]DNA polymerase eta [Homo sapiens] [gi:5729982]
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2
[SID50105803]
Potency 1.4125qHTS Assay for Inhibitors of DNA Polymerase Beta [AID485314, Type: confirmatory]DNA polymerase beta [Homo sapiens] [gi:4505931]
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3
[SID50105803]
Potency 2.2387qHTS for Inhibitors of Polymerase Iota [AID588590, Type: confirmatory]DNA polymerase iota [Homo sapiens] [gi:154350220]
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4
[SID11110721]
Potency 2.5119qHTS Assay for Inhibitors of 15-hLO (15-human lipoxygenase) [AID887, Type: confirmatory]15-lipoxygenase [Homo sapiens] [gi:1832253]
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5
[SID50105803]
Potency 3.5481qHTS Assay for Inhibitors of RecQ-Like Dna Helicase 1 (RECQ1) [AID2549, Type: confirmatory]Chain A, Structure Of Human Recq-Like Helicase In Complex With A Dna Substrate [gi:282403581]
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6
[SID50105803]
Potency 3.9811qHTS Validation Assay for Inhibitors of RecQ-Like Dna Helicase 1 (RECQ1) [AID2353, Type: confirmatory]Chain A, Structure Of Human Recq-Like Helicase In Complex With A Dna Substrate [gi:282403581]
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7
[SID90341148]
Potency 6.3096qHTS Assay for Inhibitors of GCN5L2 [AID504327, Type: confirmatory]histone acetyltransferase KAT2A [Homo sapiens] [gi:153791535]
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8
[SID103410804]
IC50 7Inhibition of fatty acid amide hydrolase; range = 4.1-7 uM [AID242030, Type: Literature]
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9
[SID90341148]
Potency 7.5193qHTS for Inhibitors of Polymerase Kappa [AID588579, Type: confirmatory]DNA polymerase kappa [Homo sapiens] [gi:7705344]
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10
[SID11110721]
Potency 7.9433qHTS Assay for Inhibitors of HSD17B4, hydroxysteroid (17-beta) dehydrogenase 4 [AID893, Type: confirmatory]Chain B, The Structure Of Wild-Type Human Hadh2 (17beta-Hydroxysteroid Dehydrogenase Type 10) Bound To Nad+ At 1.2 A [gi:122921311]
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11
[SID11110721]
Potency 7.9433qHTS Assay for Inhibitors of HSD17B4, hydroxysteroid (17-beta) dehydrogenase 4 [AID893, Type: confirmatory]Chain A, The Structure Of Wild-Type Human Hadh2 (17beta-Hydroxysteroid Dehydrogenase Type 10) Bound To Nad+ At 1.2 A [gi:122921310]
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12
[SID11110721]
Potency 10qHTS Assay for Inhibitors of 15-hLO-2 (15-human lipoxygenase 2) [AID881, Type: confirmatory]Arachidonate 15-lipoxygenase B [gi:317373425]
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13
[SID90341148]
Potency 11.9173qHTS Assay for Inhibitors of Histone Lysine Methyltransferase G9a [AID504332, Type: confirmatory]euchromatic histone-lysine N-methyltransferase 2 [Homo sapiens] [gi:168985070]
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14
[SID103410804]
IC50 12.5892Antiplasmodial activity against Plasmodium falciparum HB3 after 72 hrs by SYBR green assay [AID524795, Type: Literature]
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15
[SID103410804]
IC50 12.5892Antiplasmodial activity against Plasmodium falciparum 7G8 after 72 hrs by SYBR green assay [AID524791, Type: Literature]
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16
[SID103410804]
IC50 12.5892Antiplasmodial activity against Plasmodium falciparum D10 after 72 hrs by SYBR green assay [AID524792, Type: Literature]
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17
[SID50105803]
Potency 14.1254qHTS for differential inhibitors of proliferation of Plasmodium falciparum line HB3 [AID1886, Type: confirmatory]
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18
[SID50105803]
Potency 14.1254qHTS for differential inhibitors of proliferation of Plasmodium falciparum line 7G8 [AID1815, Type: confirmatory]
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19
[SID50105803]
Potency 14.1254qHTS for differential inhibitors of proliferation of Plasmodium falciparum line GB4 [AID1816, Type: confirmatory]
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20
[SID103410804]
IC50 15.8489Antiplasmodial activity against Plasmodium falciparum W2 after 72 hrs by SYBR green assay [AID524796, Type: Literature]
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21
[SID103410804]
IC50 15.8489Antiplasmodial activity against Plasmodium falciparum 3D7 after 72 hrs by SYBR green assay [AID524790, Type: Literature]
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22
[SID103410804]
IC50 15.8489Antiplasmodial activity against Plasmodium falciparum GB4 after 72 hrs by SYBR green assay [AID524794, Type: Literature]
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23
[SID50105803]
Potency 17.7828qHTS Assay for Inhibitors of Influenza NS1 Protein Function [AID2326, Type: confirmatory]nonstructural protein 1 [Influenza A virus (A/WSN/1933(H1N1))] [gi:194352380]
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24
[SID90341148]
Potency 18.8876Inhibitors of USP1/UAF1: Pilot qHTS [AID504865, Type: confirmatory]USP1 protein [Homo sapiens] [gi:118600387]
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25
[SID50105803]
Potency 22.3872qHTS Assay for Inhibitors of Human Jumonji Domain Containing 2E (JMJD2E) [AID2147, Type: confirmatory]Chain A, Crystal Structure Of The Human 2-Oxoglutarate Oxygenase Loc390245 [gi:221046486]
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26
[SID50105803]
Potency 28.1838Confirmation Assay for Inhibitors of Tyrosyl-DNA Phosphodiesterase (TDP1) [AID489007, Type: confirmatory]Chain A, Crystal Structure Of Human Tyrosyl-Dna Phosphodiesterase (Tdp1) [gi:20150581]
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27
[SID50105803]
Potency 28.1838qHTS Validation Assay for Inhibitors of the Human Apurinic/apyrimidinic Endonuclease 1 (APE1) [AID1705, Type: confirmatory]Chain A, Human Ape1 Endonuclease With Bound Abasic Dna And Mn2+ Ion [gi:6980812]
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28
[SID26753515]
Potency 28.1838qHTS Assay for Inhibitors of HPGD (15-Hydroxyprostaglandin Dehydrogenase) [AID894, Type: confirmatory]15-hydroxyprostaglandin dehydrogenase [NAD(+)] isoform 1 [Homo sapiens] [gi:31542939]
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29
[SID170466894]
Potency-Replicate_1 29.847qHTS assay to identify small molecule agonists of the farnesoid-X-receptor (FXR) signaling pathway - cell viability counter screen [AID743218, Type: confirmatory]
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30
[SID50105803]
Potency 31.6228qHTS Assay for Inhibitors of Tyrosyl-DNA Phosphodiesterase (TDP1) [AID485290, Type: confirmatory]Chain A, Crystal Structure Of Human Tyrosyl-Dna Phosphodiesterase (Tdp1) [gi:20150581]
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31
[SID90341148]
Potency 39.8107Inhibitors of the vitamin D receptor (VDR): qHTS [AID504847, Type: confirmatory]vitamin D3 receptor isoform VDRA [Homo sapiens] [gi:63054845]
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32
[SID90341148]
Potency 44.6684qHTS Validation Assay for Inhibitors of HP1-beta Chromodomain Interactions with Methylated Histone Tails [AID488953, Type: confirmatory]chromobox protein homolog 1 [Homo sapiens] [gi:187960037]
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33
[SID26753515]
Potency 79.4328qHTS Assay for Inhibitors of Bacillus subtilis Sfp phosphopantetheinyl transferase (PPTase) [AID1490, Type: confirmatory]phosphopantetheinyl transferase [Bacillus subtilis] [gi:10954339]
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34
[SID103410804]
Ki 10In vitro binding affinity was determined against rat brain Cannabinoid receptor 1 [AID49668, Type: Literature]
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35
[SID11110721]
Cytochrome panel assay with activity outcomes [AID1851, Type: other]
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36
[SID104171102]
qHTS profiling for inhibitors of Plasmodium falciparum proliferation [AID504749, Type: Literature]
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37
[SID103410804]
Antiinflammatory activity in TNFalpha-stimulated mouse RAW264.7 cells assessed as PGJ level at 1 uM after 20 hrs by ELISA [AID639998, Type: Literature]
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38
[SID103410804]
Antiinflammatory activity in TNFalpha-stimulated mouse RAW264.7 cells assessed as PGJ level at 10 uM after 20 hrs by ELISA [AID640001, Type: Literature]
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39
[SID103410804]
Ratio of iPGJ2 to iPGE in LPS-induced mouse RAW264.7 cells at 1 uM by ELISA [AID287976, Type: Literature]
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40
[SID103410804]
Reduction of phorbol ester-induced ear edema in CD1 mouse assessed as ear thickness at 200 ug/ear [AID287977, Type: Literature]
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41
[SID103410804]
Antiproliferative activity against rat RBL2H3 cells at 0.1 uM treated 1 hr before LPS-challenge assessed after 24 hrs relative to control [AID387969, Type: Literature]
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42
[SID103410804]
Antiproliferative activity against rat RBL2H3 cells at 1 uM treated 1 hr before LPS-challenge assessed after 24 hrs relative to control [AID387970, Type: Literature]
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43
[SID103410804]
Antiproliferative activity against rat RBL2H3 cells at 10 uM treated 1 hr before LPS-challenge assessed after 24 hrs relative to control [AID387971, Type: Literature]
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44
[SID26753513]
qHTS profiling for inhibitors of Plasmodium falciparum proliferation [AID504749, Type: Literature]
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45
[SID103410804]
Antiproliferative activity against LPS-induced mouse RAW264.7 cells assessed as number of cells at 10 uM after 48 hrs [AID287964, Type: Literature]
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46
[SID103410804]
Effect on iPGE2 level in LPS-induced mouse RAW264.7 cells at 10 uM by ELISA [AID287966, Type: Literature]
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47
[SID103410804]
Effect on iPGE2 level in LPS-induced mouse RAW264.7 cells at 1 uM by ELISA [AID287968, Type: Literature]
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48
[SID103410804]
Effect on iPGJ2 level in LPS-induced mouse RAW264.7 cells at 10 uM by ELISA [AID287970, Type: Literature]
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49
[SID103410804]
Effect on iPGJ2 level in LPS-induced mouse RAW264.7 cells at 1 uM by ELISA [AID287972, Type: Literature]
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50
[SID103410804]
Ratio of iPGJ2 to iPGE in LPS-induced mouse RAW264.7 cells at 10 uM by ELISA [AID287974, Type: Literature]
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