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Thromboxane B2 (CID 5283137) - Compound BioActivity Data
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BioActivity Outcomes:
Inactive(39)
 
 
Inconclusive(2)
 
 
Unspecified(9)
 
 
Top Targets:
KAZAL SLC21(5)
 
 
ABCC MRP doma..(3)
 
 
NR LBD ROR li..(2)
 
 
HELICc(2)
 
 
PLN02808(2)
 
 
BioAssay Types:
Confirmatory(39)
 
 
 
Literature(9)
 
 
Screening(2)
 
 
BioActivity Types:
Potency(36)
 
 
 
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 47    Data Row: 50   Total Pages: 3   Display: Page     
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#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID160693341]
Km 0.423TP_TRANSPORTER: uptake in PGT-expressing HeLa cells [AID681576, Type: Literature]Solute carrier organic anion transporter family member 2A1 [gi:357529156]
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2
[SID160693341]
TP_TRANSPORTER: inhibition of alaninyl-d4TMP by Thromboxane B2 at a concentration of 20uM in membrane vesicle from MRP5-expressing HEK293 cells [AID681870, Type: Literature]Multidrug resistance-associated protein 5 [gi:8928547]
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3
[SID160693341]
Km TP_TRANSPORTER: uptake in Xenopus laevis oocytes [AID681342, Type: Literature]Solute carrier organic anion transporter family member 1B1 [gi:12643959]
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4
[SID160693341]
Km TP_TRANSPORTER: uptake in Xenopus laevis oocytes [AID681173, Type: Literature]Solute carrier organic anion transporter family member 2B1 [gi:27734548]
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5
[SID160693341]
TP_TRANSPORTER: inhibition of alaninyl-d4TMP by Thromboxane B2 at a concentration of 20uM in membrane vesicle from MRP3-expressing Sf9 cells [AID680416, Type: Literature]Multidrug resistance associated protein [gi:74761045]
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6
[SID160693341]
TP_TRANSPORTER: inhibition of alaninyl-d4TMP in the presence of Thromboxane B2 at a concentration of 20uM in membrane vesicles from MRP4-expressing Sf9 cells [AID681886, Type: Literature]Multidrug resistance-associated protein 4 [gi:206729914]
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7
[SID160693341]
TP_TRANSPORTER: uptake in PGT-expressing HeLa cells [AID682149, Type: Literature]Solute carrier organic anion transporter family member 2A1 [gi:218511799]
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8
[SID160693341]
TP_TRANSPORTER: inhibition of alaninyl-d4TMP in the presence of Thromboxane B2 at a concentration of 20uM in membrane vesicles from MRP1-expressing Sf9 cells [AID681092, Type: Literature]Multidrug resistance-associated protein 1 [gi:296439301]
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9
[SID160693341]
Km TP_TRANSPORTER: uptake in Xenopus laevis oocytes [AID681367, Type: Literature]Solute carrier organic anion transporter family member 3A1 [gi:296452954]
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10
[SID26754848]
Potency qHTS Assay for Inhibitors Targeting the Menin-MLL Interaction in MLL Related Leukemias: Competition With Fluorescein Labeled MLL-derived Peptide [AID1766, Type: confirmatory]histone-lysine N-methyltransferase 2A isoform 2 precursor [Homo sapiens] [gi:56550039]
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11
[SID26754848]
Potency Inhibitors of the vitamin D receptor (VDR): qHTS [AID504847, Type: confirmatory]vitamin D3 receptor isoform VDRA [Homo sapiens] [gi:63054845]
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12
[SID26754848]
Potency qHTS Assay for Inhibitors of the ERK Signaling Pathway using a Homogeneous Screening Assay; Stimulation with EGF [AID1454, Type: confirmatory]mitogen-activated protein kinase 1 [Homo sapiens] [gi:66932916]
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13
[SID26754848]
Potency qHTS Assay for Inhibitors of Human Jumonji Domain Containing 2E (JMJD2E) [AID2147, Type: confirmatory]Chain A, Crystal Structure Of The Human 2-Oxoglutarate Oxygenase Loc390245 [gi:221046486]
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14
[SID26754848]
Potency qHTS Assay for Promiscuous and Specific Inhibitors of Cruzain (with detergent) [AID1478, Type: confirmatory]Chain A, Crystal Structure Of Cruzain Covalently Bound To A Purine Nitrile [gi:281307097]
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15
[SID26754848]
Potency qHTS Assay for Promiscuous and Specific Inhibitors of Cruzain (without detergent) [AID1476, Type: confirmatory]Chain A, Crystal Structure Of Cruzain Covalently Bound To A Purine Nitrile [gi:281307097]
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16
[SID26754848]
Potency qHTS Assay for Inhibitors of RecQ-Like Dna Helicase 1 (RECQ1) [AID2549, Type: confirmatory]Chain A, Structure Of Human Recq-Like Helicase In Complex With A Dna Substrate [gi:282403581]
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17
[SID26754848]
qHTS Multiplex Assay to Identify Dual Action Probes in a Cell Model of Huntington: Cytoprotection (ATP) [AID1471, Type: confirmatory]huntingtin [Homo sapiens] [gi:90903231]
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18
[SID26754848]
Potency qHTS for Inhibitors of Tau Fibril Formation, Thioflavin T Binding [AID1460, Type: confirmatory]Microtubule-associated protein tau [Homo sapiens] [gi:92096784]
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19
[SID26754848]
Potency qHTS for Inhibitors of Tau Fibril Formation, Fluorescence Polarization [AID1468, Type: confirmatory]Microtubule-associated protein tau [Homo sapiens] [gi:92096784]
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20
[SID26754848]
Potency qHTS Assay for Inhibitors and Activators of Human alpha-Glucosidase From Spleen Homogenate [AID2112, Type: confirmatory]lysosomal alpha-glucosidase preproprotein [Homo sapiens] [gi:119393891]
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