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tectochrysin (CID 5281954) - Compound BioActivity Data
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BioActivity Outcomes:
Active(19)
 
 
Inactive(773)
 
 
Inconclusive(22)
 
 
Unspecified(40)
 
 
Top Targets:
7TM GPCR Srx(24)
 
 
7TM GPCR Srsx(17)
 
 
PAS(11)
 
 
 
 
Bcl-2 like(11)
 
 
alkPPc(10)
 
 
BioAssay Types:
Screening(479)
 
 
 
 
Confirmatory(279)
 
 
 
 
 
Literature(72)
 
 
 
 
BioActivity Types:
Potency(202)
 
 
 
 
 
IC50(42)
 
 
 
EC50(13)
 
 
 
Kd(2)
 
 
AC50(1)
 
 
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 747    Data Row: 854   Total Pages: 43   Display: Page     
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#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID11113093]
Potency 0.3981qHTS Assay for Inhibitors and Substrates of Cytochrome P450 2C19 [AID899, Type: confirmatory]cytochrome P450 2C19 precursor [Homo sapiens] [gi:4503219]
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2
[SID103418563]
Kd 6.3Effect of Chrysin Alkylation on the Binding to PgP Cytosolic Domain. [AID27150, Type: Literature]
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3
[SID103418563]
Kd 6.30957Binding affinity to ABCB1 nucleotide binding domain 2 [AID615921, Type: Literature]
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4
[SID26754333]
Potency 10qHTS Assay for Inhibitors and Substrates of Cytochrome P450 3A4 [AID884, Type: confirmatory]cytochrome P450 3A4 isoform 1 [Homo sapiens] [gi:13435386]
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5
[SID26725301]
AbsAC40_uM 14.179MITF Measured in Cell-Based System Using Plate Reader - 2084-01_Activator_Dose_CherryPick_Activity [AID540258, Type: confirmatory]
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6
[SID103418563]
IC50 23Inhibition of LPS-induced NO production in ddY mouse macrophages assessed as nitrate accumulation after 20 hrs by Griess reagent method [AID358994, Type: Literature]
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7
[SID26725301]
AC50_uM 46.163MITF Act Counter Assay: HeLa CTG Assay Measured in Cell-Based System Using Plate Reader - 2084-08_Activator_Dose_CherryPick_Activity [AID540259, Type: confirmatory]
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8
[SID103418563]
IC50 49Inhibition of rat RBL2H3 cell degranulation assessed as inhibition of beta-hexosamidase release after 10 mins by microplate reader assay [AID359218, Type: Literature]
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9
[SID26725301]
MITF Measured in Cell-Based System Using Plate Reader - 2084-01_Activator_SinglePoint_HTS_Activity [AID588334, Type: screening]
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10
[SID24824136]
MLPCN Alpha-Synuclein 5'UTR - 5'-UTR binding - activators [AID1814, Type: screening]
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11
[SID24824136]
Cycloheximide Counterscreen for Small Molecule Inhibitors of Shiga Toxin [AID2314, Type: screening]shiga toxin 1 variant A subunit [Escherichia coli O157:H7] [gi:32400299]
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12
[SID11113093]
p450-cyp1a2 [AID410, Type: confirmatory]cytochrome P450 1A2 [Homo sapiens] [gi:73915100]
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13
[SID103418563]
Effect on AhR-mediated CYP1A1 activation in mouse Hepa1c1c12 cells at 20 uM after 18 hrs by Western blot analysis [AID431868, Type: Literature]Aryl hydrocarbon receptor [gi:29337198]
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14
[SID103418563]
Effect on AhR-mediated NAPDH quinine reductase activation in mouse Hepa1c1c12 cells at 20 uM after 18 hrs by Western blot analysis [AID431869, Type: Literature]Aryl hydrocarbon receptor [gi:29337198]
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15
[SID103418563]
Induction of nuclear translocation of AhR from cytosol in mouse Hepa1 cells at 20 uM after 60 mins using DAPI staining by microscopic analysis [AID431870, Type: Literature]Aryl hydrocarbon receptor [gi:29337198]
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16
[SID24824136]
Cycloheximide Counterscreen for Small Molecule Inhibitors of Shiga Toxin [AID2314, Type: screening]shiga toxin 1 B subunit [Escherichia coli O157:H7] [gi:32400300]
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17
[SID11113093]
qHTS Assay for Tau Filament Binding [AID596, Type: confirmatory]Microtubule-associated protein tau [Homo sapiens] [gi:92096784]
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18
[SID26725301]
uHTS Fluorescent Assay Using Nedd8 Protein Substrate for Identification of Inhibitors of Sentrin-Specific Protease 8 (SENP8) [AID602440, Type: screening]sentrin-specific protease 8 [Homo sapiens] [gi:262118306]
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19
[SID26725301]
Screen for inhibitors of the SWI/SNF chromatin remodeling complex (esBAF) in mouse embryonic stem cells with Luciferase reporter assay Measured in Cell-Based System Using Plate Reader - 2141-01_Inhibitor_SinglePoint_HTS_Activity [AID602393, Type: screening]transcription activator BRG1 isoform 1 [Mus musculus] [gi:291463269]
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20
[SID11113093]
Potency 31.6228qHTS Assay for Agonists of the Thyroid Stimulating Hormone Receptor [AID926, Type: confirmatory]thyroid stimulating hormone receptor [Homo sapiens] [gi:38016895]
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