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3-methylquercetin (CID 5281654) - Compound BioActivity Data
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BioActivity Outcomes:
Active(19)
 
 
Inactive(73)
 
 
Inconclusive(13)
 
 
Unspecified(27)
 
 
Top Targets:
NR LBD ROR li..(4)
 
 
SLT beta(4)
 
 
 
Bromo ALL-1(4)
 
 
 
HELICc(4)
 
 
Menin(4)
 
 
 
BioAssay Types:
Confirmatory(61)
 
 
 
 
Literature(47)
 
 
 
 
 
Screening(24)
 
 
 
BioActivity Types:
Potency(61)
 
 
 
 
IC50(20)
 
 
 
 
Ki(1)
 
 
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 101    Data Row: 132   Total Pages: 7   Display: Page     
Sort: [Click the result table header to sort]
#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID103489401]
IC50 0.017Inhibition of human CYP1B1 by EROD assay [AID502475, Type: Literature]Cytochrome P450 1B1 [gi:48429256]
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2
[SID103489401]
IC50 0.056Inhibition of human CYP1A1 by EROD assay [AID502474, Type: Literature]Cytochrome P450 1A1 [gi:117139]
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3
[SID103489401]
IC50 0.5Inhibition of CK2 assessed as level of ATP utilized by luciferase-based bioluminescence assay [AID353598, Type: Literature]
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4
[SID103489401]
IC50 0.91Inhibition of CAMK2 assessed as level of ATP utilized by luciferase-based bioluminescence assay [AID353599, Type: Literature]
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5
[SID103489401]
IC50 1.261Inhibition of human CYP1A2 by EROD assay [AID502473, Type: Literature]Cytochrome P450 1A2 [gi:117144]
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6
[SID103489401]
IC50 2.51Inhibition of xanthine oxidase assessed as decrease in uric acid production by spectrophotometry [AID399340, Type: Literature]
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7
[SID103489401]
IC50 2.75Antioxidant activity assessed as superoxide-scavenging activity by nitrite method [AID399341, Type: Literature]
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8
[SID103489401]
IC50 3.8Inhibition of procoagulant activity in monocyte from human blood assessed as counteraction of IL1-induced tissue factor expression after 18 hrs [AID400608, Type: Literature]
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9
[SID103489401]
IC50 5Inhibition of FabI [AID265759, Type: Literature]Enoyl-acyl-carrier protein reductase precursor [gi:74844868]
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10
[SID103489401]
IC50 8.3Inhibition of FabG [AID265760, Type: Literature]3-oxoacyl-acyl-carrier protein reductase precursor [gi:75020671]
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11
[SID103489401]
IC50 14.7Antiplasmodial activity against chloroquine-sensitive Plasmodium falciparum NF54 [AID265761, Type: Literature]
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12
[SID85843252]
Luminescence Homogenous Primary HTS to Identify Inhibitors of STK33 Activity [AID2322, Type: screening]
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13
[SID103489401]
Inhibition of heat-induced HSP70 expression in human Jurkat cells at 50 ug/mL treated for 1 hr before heat induction by Western blot [AID353590, Type: Literature]
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14
[SID26756953]
Cycloheximide Counterscreen for Small Molecule Inhibitors of Shiga Toxin [AID2314, Type: screening]shiga toxin 1 B subunit [Escherichia coli O157:H7] [gi:32400300]
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15
[SID26756952]
A qHTS for Small Molecule Inhibitors of Shiga Toxin [AID2315, Type: screening]shiga toxin 1 B subunit [Escherichia coli O157:H7] [gi:32400300]
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16
[SID26756953]
A qHTS for Small Molecule Inhibitors of Shiga Toxin [AID2315, Type: screening]shiga toxin 1 B subunit [Escherichia coli O157:H7] [gi:32400300]
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17
[SID26756953]
Cycloheximide Counterscreen for Small Molecule Inhibitors of Shiga Toxin [AID2314, Type: screening]shiga toxin 1 variant A subunit [Escherichia coli O157:H7] [gi:32400299]
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18
[SID26756952]
A qHTS for Small Molecule Inhibitors of Shiga Toxin [AID2315, Type: screening]shiga toxin 1 variant A subunit [Escherichia coli O157:H7] [gi:32400299]
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19
[SID26756953]
A qHTS for Small Molecule Inhibitors of Shiga Toxin [AID2315, Type: screening]shiga toxin 1 variant A subunit [Escherichia coli O157:H7] [gi:32400299]
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20
[SID103489401]
IC50 10Cytotoxicity against human HeLa cells by MTT assay [AID423636, Type: Literature]
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