Bookmark and Share
isoquercitrin (CID 5280804) - Compound BioActivity Data
.
BioActivity Outcomes:
Active(70)
 
 
Inactive(320)
 
 
Inconclusive(9)
 
 
Unspecified(156)
 
 
Top Targets:
7tm 4(20)
 
 
 
 
alkPPc(19)
 
 
 
Bcl-2 like(9)
 
 
M2 ACE(7)
 
 
NR LBD PPAR(7)
 
 
 
BioAssay Types:
Literature(232)
 
 
 
 
 
Screening(189)
 
 
 
 
Confirmatory(110)
 
 
 
 
 
BioActivity Types:
IC50(62)
 
 
 
 
Potency(58)
 
 
 
 
EC50(18)
 
 
 
 
Ki(1)
 
 
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 522    Data Row: 555   Total Pages: 28   Display: Page     
Sort: [Click the result table header to sort]
#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID103557565]
ED50 1.2Antiviral activity against influenza A virus (A/swine/OH/511445/2007(H1N1)) Oh7 infected in MDCK cells assessed as inhibition of viral replication after 4 days by quantitative RT-PCR [AID638568, Type: Literature]
View
2
[SID49681636]
IC50_Mean 1.66Dose Response confirmation of uHTS hits from a small molecule inhibitors of mouse intestinal alkaline phosphatase via a luminescent assay [AID488785, Type: confirmatory]intestinal alkaline phosphatase precursor [Mus musculus] [gi:124487323]
View
3
[SID26719900]
Potency 1.7783qHTS Assay for Inhibitors of DNA Polymerase Beta [AID485314, Type: confirmatory]DNA polymerase beta [Homo sapiens] [gi:4505931]
View
4
[SID103557565]
IC50 2Inhibition of Leishmania amazonensis recombinant arginase expressed in Escherichia coli Rosetta (DE3) pLysS using L-arginine as substrate incubated for 10 mins prior to substrate addition measured after 10 mins by colorimetry [AID1066694, Type: Literature]Arginase [gi:74764753]
View
5
[SID26719900]
Potency 3.5481qHTS Assay for Inhibitors and Activators of Human alpha-Glucosidase Cleavage of Glycogen [AID2100, Type: confirmatory]lysosomal alpha-glucosidase preproprotein [Homo sapiens] [gi:119393891]
View
6
[SID103557565]
IC50 4.05Antiplasmodial activity against chloroquine-resistant blood stage Plasmodium falciparum Dd2 after 72 hrs by SYBR Green I-based fluorescence assay [AID1072080, Type: Literature]
View
7
[SID103557565]
IC50 4.4Inhibition of Sprague-Dawley rat lens aldose reductase [AID654333, Type: Literature]Aldose reductase [gi:1168407]
View
8
[SID103557565]
IC50 4.5Inhibition of human recombinant aldose reductase using D-glyceraldehyde as substrate preincubated for 10 mins before substrate addition measured for every 10 secs for 50 mins by spectrophotometry [AID639825, Type: Literature]Aldose reductase [gi:113596]
View
9
[SID49681636]
IC50_Mean 5.25Dose Response confirmation of uHTS hits from a small molecule inhibitors of human intestinal alkaline phosphatase via a luminescent assay [AID463135, Type: confirmatory]Alkaline phosphatase, intestinal [Homo sapiens] [gi:124376142]
View
10
[SID103557565]
IC50 5.54Antiplasmodial activity against chloroquine-sensitive blood stage Plasmodium falciparum 3D7 after 72 hrs by SYBR Green I-based fluorescence assay [AID1072081, Type: Literature]
View
11
[SID26719900]
Potency 8.9125qHTS Assay for Inhibitors of Histone Lysine Methyltransferase G9a [AID504332, Type: confirmatory]euchromatic histone-lysine N-methyltransferase 2 [Homo sapiens] [gi:168985070]
View
12
[SID49681636]
IC50_Mean 8.96Dose Response confirmation of uHTS inhibitors of Mouse Intestinal Alkaline Phosphatase using Human Intestinal Alkaline Phosphatase [AID488876, Type: confirmatory]Alkaline phosphatase, intestinal [Homo sapiens] [gi:124376142]
View
13
[SID103557565]
IC50 9.2Inhibition of advanced glycation end-products formation after 14 days by spectrofluorimetry [AID654332, Type: Literature]
View
14
[SID103557565]
IC50 10.28Inhibition of CDK5/p25 (unknown origin) after 30 mins by SDS-PAGE analysis [AID767308, Type: Literature]Cyclin-dependent kinase 5 [gi:4033704]
View
15
[SID103557565]
IC50 10.28Inhibition of CDK5/p25 (unknown origin) after 30 mins by SDS-PAGE analysis [AID767308, Type: Literature]Cyclin-dependent kinase 5 activator 1 [gi:2498217]
View
16
[SID103557565]
IC50 11.7Antioxidant activity assessed as DPPH radical scavenging activity after 10 mins [AID597947, Type: Literature]
View
17
[SID26719900]
Potency 12.5893qHTS Assay for Inhibitors of Human Jumonji Domain Containing 2E (JMJD2E) [AID2147, Type: confirmatory]Chain A, Crystal Structure Of The Human 2-Oxoglutarate Oxygenase Loc390245 [gi:221046486]
View
18
[SID49681636]
IC50_Mean 14Dose Response confirmation of uHTS inhibitors of Mouse Intestinal Alkaline Phosphatase using Tissue Nonspecific Alkaline Phosphatase. [AID488906, Type: confirmatory]alkaline phosphatase, tissue-nonspecific isozyme isoform 1 precursor [Homo sapiens] [gi:116734717]
View
19
[SID103557565]
IC50 15.74Inhibition of recombinant Plasmodium falciparum falcipain 2 after 30 mins by fluorescence assay [AID1072082, Type: Literature]
View
20
[SID49681636]
EC50_uM 15.8Luminescence Cell-Free Homogeneous Dose Retest to Identify Inhibitors of Glycogen Synthase Kinase-3 beta Activity [AID434954, Type: confirmatory]glycogen synthase kinase-3 beta isoform 1 [Homo sapiens] [gi:21361340]
View