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BioActivity Data for Compound Quercetin (CID 5280343)

BioActivity Outcomes:
Active(633)
 
 
Inactive(748)
 
 
Inconclusive(247)
 
 
Unspecified(783)
 
 
Top Targets:
p450(29)
 
 
 
 
 
Tryp SPc(24)
 
 
 
 
NR LBD TR(20)
 
 
 
 
NR LBD PPAR(19)
 
 
 
 
 
NR LBD GR(18)
 
 
 
 
BioAssay Types:
Literature(1325)
 
 
 
 
 
Confirmatory(805)
 
 
 
 
 
Screening(65)
 
 
 
Summary(59)
 
 
 
 
BioAssay Categories:
In vitro(68)
 
 
 
 
 
In vivo(24)
 
 
 
 
 
Biochemical(525)
 
 
 
 
 
Toxicity(129)
 
 
 
 
 
ADME(114)
 
 
 
 
 
Cell-based(381)
 
 
 
 
 
Organism-base..(2)
 
 
BioActivity Types:
Potency(680)
 
 
 
 
 
IC50(360)
 
 
 
 
 
EC50(46)
 
 
 
Ki(46)
 
 
 
 
Kd(5)
 
 
 
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 1910    Data Row: 2411   Total Pages: 121   Display: Page     
Sort: [Click the result table header to sort]
#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID103167027]
IC50 0.01Inhibition of bovine MAO-A by fluorimetric method [AID377654, Type: Literature]Amine oxidase [flavin-containing] A [gi:124028637]
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2
[SID103167027]
IC50 0.012Inhibition of human placental microsome CYP19 [AID479369, Type: Literature]Aromatase [gi:117293]
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3
[SID103167027]
IC50 0.0148Inhibition of cataracted human eye lens aldose reductase [AID388742, Type: Literature]Aldose reductase [gi:113596]
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4
[SID103167027]
Ki 0.022Inhibition of Plasmodium falciparum ENR in presence of triclosan [AID277587, Type: Literature]Enoyl-acyl-carrier protein reductase precursor [gi:74844868]
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5
[SID103167027]
Ki 0.023Inhibition of CYP1B1 EROD activity assessed as inhibition of deethylation of 7-ethoxyresorufin to resorufin [AID598342, Type: Literature]
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6
[SID103167027]
Kd 0.0387Inhibition of human thrombin assessed as equilibrium dissociation constant at 50 to 1000 uM by BIAcore analysis [AID768894, Type: Literature]Prothrombin [gi:135807]
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7
[SID103167027]
IC50 0.043Inhibitory activity against PIM1 [AID257081, Type: Literature]Serine/threonine-protein kinase pim-1 [gi:83305339]
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8
[SID103167027]
Ki 0.0453Inhibition of rat ecto-5'-nucleotidase expressed in Sf9 cells by capillary electrophoresis method [AID461575, Type: Literature]5'-nucleotidase [gi:112826]
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9
[SID103167027]
IC50 0.06Antioxidant activity assessed as scavenging of glucose oxidase-generated H2O2 and hydroxyl radicals by chemiluminescence assay [AID710235, Type: Literature]
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10
[SID103167027]
IC50 0.077Inhibition of human CYP1B1 by EROD assay [AID502475, Type: Literature]Cytochrome P450 1B1 [gi:48429256]
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11
[SID103167027]
IC50 0.12Inhibition of SRC (unknown origin) [AID1063039, Type: Literature]Proto-oncogene tyrosine-protein kinase Src [gi:125711]
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12
[SID11111705]
Potency 0.1259qHTS Assay for Inhibitors of HADH2 (Hydroxyacyl-Coenzyme A Dehydrogenase, Type II) [AID886, Type: confirmatory]Chain A, The Structure Of Wild-Type Human Hadh2 (17beta-Hydroxysteroid Dehydrogenase Type 10) Bound To Nad+ At 1.2 A [gi:122921310]
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13
[SID11111705]
Potency 0.1259qHTS Assay for Inhibitors of HADH2 (Hydroxyacyl-Coenzyme A Dehydrogenase, Type II) [AID886, Type: confirmatory]Chain B, The Structure Of Wild-Type Human Hadh2 (17beta-Hydroxysteroid Dehydrogenase Type 10) Bound To Nad+ At 1.2 A [gi:122921311]
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14
[SID103167027]
IC50 0.14Inhibition of Escherichia coli DNA gyrase assessed as inhibition of pBR322 supercoiling by densitometry [AID603461, Type: Literature]
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15
[SID103167027]
I50 0.145Inhibition of beef heart mitochondrial NADH oxidase assessed per mg of protein [AID338027, Type: Literature]
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16
[SID11111706]
Potency 0.1585qHTS Assay for Inhibitors of HADH2 (Hydroxyacyl-Coenzyme A Dehydrogenase, Type II) [AID886, Type: confirmatory]Chain B, The Structure Of Wild-Type Human Hadh2 (17beta-Hydroxysteroid Dehydrogenase Type 10) Bound To Nad+ At 1.2 A [gi:122921311]
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17
[SID11111706]
Potency 0.1585qHTS Assay for Inhibitors of HADH2 (Hydroxyacyl-Coenzyme A Dehydrogenase, Type II) [AID886, Type: confirmatory]Chain A, The Structure Of Wild-Type Human Hadh2 (17beta-Hydroxysteroid Dehydrogenase Type 10) Bound To Nad+ At 1.2 A [gi:122921310]
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18
[SID103167027]
ID50 0.17Inhibition of Moloney murine leukemia virus reverse transcriptase using (ribocytidylic acid)n(deoxyguanylic acid)12-18 as template primer by liquid scintillation counting [AID339057, Type: Literature]
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19
[SID50104737]
Potency 0.1995qHTS Assay for Inhibitors of DNA Polymerase Beta [AID485314, Type: confirmatory]DNA polymerase beta [Homo sapiens] [gi:4505931]
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20
[SID124881266]
Potency 0.1995qHTS for Inhibitors of Polymerase Kappa [AID588579, Type: confirmatory]DNA polymerase kappa [Homo sapiens] [gi:7705344]
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