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Quercetin (CID 5280343) - Compound BioActivity Data
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BioActivity Outcomes:
Active(580)
 
 
Inactive(687)
 
 
Inconclusive(227)
 
 
Unspecified(650)
 
 
Top Targets:
p450(28)
 
 
 
 
 
Tryp SPc(24)
 
 
 
 
NR LBD TR(20)
 
 
 
 
NR LBD PPAR(19)
 
 
 
 
 
Tubulin-bindi..(18)
 
 
 
 
BioAssay Types:
Literature(1136)
 
 
 
 
 
Confirmatory(765)
 
 
 
 
 
Screening(65)
 
 
 
Summary(49)
 
 
 
 
BioActivity Types:
Potency(642)
 
 
 
 
 
IC50(316)
 
 
 
 
 
Ki(44)
 
 
 
 
 
EC50(34)
 
 
 
Kd(4)
 
 
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 1660    Data Row: 2144   Total Pages: 108   Display: Page     
Sort: [Click the result table header to sort]
#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID103167027]
Ki 0.0078Binding affinity to dopamine D4 receptor [AID478694, Type: Literature]
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2
[SID103167027]
IC50 0.01Inhibition of bovine MAO-A by fluorimetric method [AID377654, Type: Literature]Amine oxidase [flavin-containing] A [gi:124028637]
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3
[SID103167027]
IC50 0.012Inhibition of human placental microsome CYP19 [AID479369, Type: Literature]Aromatase [gi:117293]
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4
[SID103167027]
IC50 0.0148Inhibition of cataracted human eye lens aldose reductase [AID388742, Type: Literature]Aldose reductase [gi:113596]
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5
[SID103167027]
Ki 0.022Inhibition of Plasmodium falciparum ENR in presence of triclosan [AID277587, Type: Literature]Enoyl-acyl-carrier protein reductase precursor [gi:74844868]
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6
[SID103167027]
Ki 0.023Inhibition of CYP1B1 EROD activity assessed as inhibition of deethylation of 7-ethoxyresorufin to resorufin [AID598342, Type: Literature]
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7
[SID103167027]
Kd 0.025Binding affinity to non phosphorylated PIM1 [AID257082, Type: Literature]Serine/threonine-protein kinase pim-1 [gi:83305339]
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8
[SID103167027]
Kd 0.0387Inhibition of human thrombin assessed as equilibrium dissociation constant at 50 to 1000 uM by BIAcore analysis [AID768894, Type: Literature]Prothrombin [gi:135807]
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9
[SID103167027]
IC50 0.043Inhibitory activity against PIM1 [AID257081, Type: Literature]Serine/threonine-protein kinase pim-1 [gi:83305339]
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10
[SID103167027]
Ki 0.0453Inhibition of rat ecto-5'-nucleotidase expressed in Sf9 cells by capillary electrophoresis method [AID461575, Type: Literature]5'-nucleotidase [gi:112826]
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11
[SID103167027]
IC50 0.06Antioxidant activity assessed as scavenging of glucose oxidase-generated H2O2 and hydroxyl radicals by chemiluminescence assay [AID710235, Type: Literature]
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12
[SID103167027]
IC50 0.077Inhibition of human CYP1B1 by EROD assay [AID502475, Type: Literature]Cytochrome P450 1B1 [gi:48429256]
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13
[SID11111705]
Potency 0.1259qHTS Assay for Inhibitors of HADH2 (Hydroxyacyl-Coenzyme A Dehydrogenase, Type II) [AID886, Type: confirmatory]Chain A, The Structure Of Wild-Type Human Hadh2 (17beta-Hydroxysteroid Dehydrogenase Type 10) Bound To Nad+ At 1.2 A [gi:122921310]
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14
[SID11111705]
Potency 0.1259qHTS Assay for Inhibitors of HADH2 (Hydroxyacyl-Coenzyme A Dehydrogenase, Type II) [AID886, Type: confirmatory]Chain B, The Structure Of Wild-Type Human Hadh2 (17beta-Hydroxysteroid Dehydrogenase Type 10) Bound To Nad+ At 1.2 A [gi:122921311]
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15
[SID103167027]
IC50 0.14Inhibition of Escherichia coli DNA gyrase assessed as inhibition of pBR322 supercoiling by densitometry [AID603461, Type: Literature]
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16
[SID103167027]
IC50 0.14Inhibition of Escherichia coli DNA gyraseB assessed as inhibition of pBR322 supercoiling by densitometry [AID501421, Type: Literature]
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17
[SID103167027]
I50 0.145Inhibition of beef heart mitochondrial NADH oxidase assessed per mg of protein [AID338027, Type: Literature]
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18
[SID11111706]
Potency 0.1585qHTS Assay for Inhibitors of HADH2 (Hydroxyacyl-Coenzyme A Dehydrogenase, Type II) [AID886, Type: confirmatory]Chain B, The Structure Of Wild-Type Human Hadh2 (17beta-Hydroxysteroid Dehydrogenase Type 10) Bound To Nad+ At 1.2 A [gi:122921311]
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19
[SID11111706]
Potency 0.1585qHTS Assay for Inhibitors of HADH2 (Hydroxyacyl-Coenzyme A Dehydrogenase, Type II) [AID886, Type: confirmatory]Chain A, The Structure Of Wild-Type Human Hadh2 (17beta-Hydroxysteroid Dehydrogenase Type 10) Bound To Nad+ At 1.2 A [gi:122921310]
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20
[SID103167027]
ID50 0.17Inhibition of Moloney murine leukemia virus reverse transcriptase using (ribocytidylic acid)n(deoxyguanylic acid)12-18 as template primer by liquid scintillation counting [AID339057, Type: Literature]
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