SureCN4246800 (CID 50899554) - BioAssay Data Summary for Compound
.
BioActivity Outcomes:
Active(2)
 
 
Unspecified(2)
 
 
Top Targets:
HAD like(2)
 
 
BioAssay Types:
Literature(4)
 
 
 
BioActivity Types:
IC50(3)
 
 
 
SAR
Target summary
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Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 4    Data Row: 4   Total Pages: 1   
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#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID123094900]
IC50 0.0088Inhibition of human Ephx2 after 30 mins by fluorescence polarization assay [AID528267, Type: Literature]Bifunctional epoxide hydrolase 2 [gi:67476665]
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2
[SID123094900]
IC50 0.0088Inhibition of human Ephx2 after 30 mins by fluorescence polarization assay [AID528267, Type: Literature]Bifunctional epoxide hydrolase 2 [gi:67476665]
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3
[SID123094900]
IC50 0.083Displacement of [3H]-cDPPO from human Ephx2 by cell-based assay [AID528268, Type: Literature]Bifunctional epoxide hydrolase 2 [gi:67476665]
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4
[SID123094900]
IC50 0.083Displacement of [3H]-cDPPO from human Ephx2 by cell-based assay [AID528268, Type: Literature]Bifunctional epoxide hydrolase 2 [gi:67476665]
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5
[SID123094900]
 Metabolic stability in human liver microsomes [AID528270, Type: Literature]
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6
[SID123094900]
IC50 Inhibition of CYP3A4 [AID528269, Type: Literature]
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