CHEMBL2203532 (CID 5019834) - BioAssay Data Summary for Compound
.
BioActivity Outcomes:
Active(1)
 
 
Inactive(3)
 
 
Top Targets:
STKc AGC(2)
 
 
 
14-3-3 gamma(1)
 
 
STKc PKA(1)
 
 
BioAssay Types:
Confirmatory(3)
 
 
 
Screening(1)
 
 
BioActivity Types:
AC50(3)
 
 
 
SAR
Target summary
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 4    Data Row: 4   Total Pages: 1   
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#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID125081983]
AC50 0.977STK-33 Kinase Inhibition Measured in Biochemical System Using Plate Reader - 2052-02_Inhibitor_Dose_DryPowder_Activity_Set2 [AID588480, Type: confirmatory]serine/threonine-protein kinase 33 [Homo sapiens] [gi:23943882]
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2
[SID125081983]
AC50 0.977STK-33 Kinase Inhibition Measured in Biochemical System Using Plate Reader - 2052-02_Inhibitor_Dose_DryPowder_Activity_Set2 [AID588480, Type: confirmatory]serine/threonine-protein kinase 33 [Homo sapiens] [gi:23943882]
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3
[SID125081983]
AC50 0.977STK-33 Kinase Inhibition Measured in Biochemical System Using Plate Reader - 2052-02_Inhibitor_Dose_DryPowder_Activity_Set2 [AID588480, Type: confirmatory]serine/threonine-protein kinase 33 [Homo sapiens] [gi:23943882]
View
4
[SID125081983]
AC50 Protein Kinase A Activity Assay Measured in Biochemical System Using Plate Reader - 2052-04_Inhibitor_Dose_DryPowder_Activity_Set2 [AID588629, Type: confirmatory]cAMP-dependent protein kinase catalytic subunit alpha isoform 1 [Homo sapiens] [gi:4506055]
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5
[SID125081983]
AC50 Protein Kinase A Activity Assay Measured in Biochemical System Using Plate Reader - 2052-04_Inhibitor_Dose_DryPowder_Activity_Set2 [AID588629, Type: confirmatory]cAMP-dependent protein kinase catalytic subunit alpha isoform 1 [Homo sapiens] [gi:4506055]
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6
[SID24357786]
 HTS for 14-3-3 protein interaction modulators [AID422, Type: screening]tyrosine 3-monooxygenase/tryptophan 5-monooxygenase activation protein, gamma polypeptide [Homo sapi [gi:21464101]
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7
[SID125081983]
AC50 Counter screen for activity against Aurora B, in dose Measured in Biochemical System Using Scintillation - 2052-06_Inhibitor_Dose_DryPowder_Activity_Set3 [AID588808, Type: confirmatory]aurora kinase B [Homo sapiens] [gi:83776600]
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8
[SID125081983]
AC50 Counter screen for activity against Aurora B, in dose Measured in Biochemical System Using Scintillation - 2052-06_Inhibitor_Dose_DryPowder_Activity_Set3 [AID588808, Type: confirmatory]aurora kinase B [Homo sapiens] [gi:83776600]
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9
[SID125081983]
AC50 Counter screen for activity against Aurora B, in dose Measured in Biochemical System Using Scintillation - 2052-06_Inhibitor_Dose_DryPowder_Activity_Set3 [AID588808, Type: confirmatory]aurora kinase B [Homo sapiens] [gi:83776600]
View