Bookmark and Share
CHEMBL3099773 (CID 49837912) - Compound BioActivity Data
.
BioActivity Outcomes:
Probe(2)
 
 
Active(5)
 
 
Inactive(5)
 
 
Top Targets:
7tm 4(8)
 
 
 
 
BioAssay Types:
Confirmatory(9)
 
 
 
Summary(2)
 
 
BioActivity Types:
EC50(7)
 
 
 
IC50(2)
 
 
 
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 9    Data Row: 12   Total Pages: 1   
Sort: [Click the result table header to sort]
#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID104164387]
Summary Assay for Selective Agonists of NTR1 [AID493055, Type: summary]neurotensin receptor type 1 [Homo sapiens] [gi:110611243]
View
2
[SID126723249]
Summary Assay for Selective Agonists of NTR1 [AID493055, Type: summary]neurotensin receptor type 1 [Homo sapiens] [gi:110611243]
View
3
[SID104164387]
IC50_Mean 0.298SAR analysis of small molecule agonists of the NTR1 receptor in a dose response fluorescent-based calcium flux assay [AID602459, Type: confirmatory]neurotensin receptor type 1 [Homo sapiens] [gi:110611243]
View
4
[SID104164387]
EC50_Mean 2.01SAR analysis of small molecule Agonists NTR1 in a image based assay set 3 [AID602356, Type: confirmatory]neurotensin receptor type 1 [Homo sapiens] [gi:110611243]
View
5
[SID126723249]
EC50_Mean 4.14SAR analysis of small molecule Agonists NTR1 in a image based assay set 3 [AID602356, Type: confirmatory]neurotensin receptor type 1 [Homo sapiens] [gi:110611243]
View
6
[SID104164387]
EC50_Mean 6.1SAR analysis of small molecule agonists of the NTR1 receptor via a luminescent beta-arrestin assay [AID602427, Type: confirmatory]neurotensin receptor type 1 [Homo sapiens] [gi:110611243]
View
7
[SID104164387]
SAR analysis of small molecule agonists of the NTR1 receptor in a single concentration fluorescent-based calcium flux assay [AID602466, Type: other]neurotensin receptor type 1 [Homo sapiens] [gi:110611243]
View
8
[SID104164387]
EC50_Mean 40SAR analysis of small molecule NTR1 agonists in a image based NTR2 selectivity assay [AID588495, Type: confirmatory]neurotensin receptor type 2 [Homo sapiens] [gi:6912538]
View
9
[SID104164387]
EC50_Mean 40SAR analysis of small molecule NTR1 agonists in a image based GPR35 selectivity assay [AID588503, Type: confirmatory]G-protein coupled receptor 35 [Homo sapiens] [gi:30526188]
View
10
[SID104164387]
EC50_Mean 80SAR analysis of small molecule NTR1 agonists in a image based NTR2 selectivity assay set 2 [AID602334, Type: confirmatory]neurotensin receptor type 2 [Homo sapiens] [gi:6912538]
View
11
[SID126723249]
EC50_Mean 80SAR analysis of small molecule NTR1 agonists in a image based NTR2 selectivity assay set 2 [AID602334, Type: confirmatory]neurotensin receptor type 2 [Homo sapiens] [gi:6912538]
View
12
[SID126723249]
IC50_Mean 80SAR analysis of small molecule agonists of the NTR1 receptor via a luminescent cytotoxicity assay [AID602482, Type: confirmatory]neurotensin receptor type 1 [Homo sapiens] [gi:110611243]
View