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CHEMBL3099775 (CID 49837903) - Compound BioActivity Data
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BioActivity Outcomes:
Inactive(3)
 
 
Unspecified(2)
 
 
Top Targets:
7tm 4(4)
 
 
 
BioAssay Types:
Confirmatory(3)
 
 
Literature(2)
 
 
BioActivity Types:
EC50(4)
 
 
 
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 5    Data Row: 5   Total Pages: 1   
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#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID194180258]
EC50 56Agonist activity at NTR1 in human U2OS cells after 1 hr by beta-arrestin GFP reporter gene assay [AID1061686, Type: Literature]Neurotensin receptor type 1 [gi:62297312]
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2
[SID194180258]
Agonist activity at NTR1 in human U2OS cells after 1 hr by beta-arrestin GFP reporter gene assay relative to NT peptide [AID1061685, Type: Literature]Neurotensin receptor type 1 [gi:62297312]
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3
[SID104164396]
EC50_Mean 33SAR analysis of small molecule agonists of the NTR1 receptor via a luminescent beta-arrestin assay [AID602427, Type: confirmatory]neurotensin receptor type 1 [Homo sapiens] [gi:110611243]
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4
[SID104164396]
EC50_Mean 40SAR analysis of small molecule NTR1 agonists in a image based NTR2 selectivity assay [AID588495, Type: confirmatory]neurotensin receptor type 2 [Homo sapiens] [gi:6912538]
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5
[SID104164396]
EC50_Mean 55.8SAR analysis of small molecule Agonists NTR1 in a image based assay set 3 [AID602356, Type: confirmatory]neurotensin receptor type 1 [Homo sapiens] [gi:110611243]
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