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Phenacetin (CID 4754) - Compound BioActivity Data
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BioActivity Outcomes:
Active(10)
 
 
Inactive(1278)
 
 
Inconclusive(72)
 
 
Unspecified(1423)
 
 
Top Targets:
7tm 4(68)
 
 
 
NR LBD PPAR(34)
 
 
 
NR LBD ER(27)
 
 
 
NR LBD AR(26)
 
 
 
p450(26)
 
 
 
 
BioAssay Types:
Confirmatory(833)
 
 
 
 
 
Screening(388)
 
 
Literature(150)
 
 
 
 
 
Summary(72)
 
 
 
BioActivity Types:
Potency(669)
 
 
 
 
IC50(164)
 
 
 
 
EC50(4)
 
 
Ki(1)
 
 
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 2267    Data Row: 2783   Total Pages: 140   Display: Page     
Sort: [Click the result table header to sort]
#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID48414293]
DSSTox (CPDBAS) Carcinogenic Potency Database Summary SingleCellCall Results [AID1189, Type: other]
View
2
[SID48414293]
DSSTox (CPDBAS) Carcinogenic Potency Database Salmonella Mutagenicity [AID1194, Type: other]
View
3
[SID48414293]
DSSTox (CPDBAS) Carcinogenic Potency Database Summary Mouse Bioassay Results [AID1199, Type: other]
View
4
[SID48414293]
DSSTox (CPDBAS) Carcinogenic Potency Database Summary MultiCellCall Results [AID1205, Type: other]
View
5
[SID48414293]
DSSTox (CPDBAS) Carcinogenic Potency Database Summary Rat Bioassay Results [AID1208, Type: other]
View
6
[SID48416402]
DSSTox (FDAMDD) FDA Maximum (Recommended) Daily Dose Database [AID1195, Type: other]
View
7
[SID50086861]
Aqueous Solubility from MLSMR Stock Solutions [AID1996, Type: other]
View
8
[SID103179006]
Phospholipidosis-positive literature compound observed in rat [AID540237, Type: Literature]
View
9
[SID11112166]
Cytochrome panel assay with activity outcomes [AID1851_4, Type: other]cytochrome P450 1A2 [Homo sapiens] [gi:73915100]
View
10
[SID11112166]
p450-cyp1a2 [AID410, Type: confirmatory]cytochrome P450 1A2 [Homo sapiens] [gi:73915100]
View
11
[SID103179006]
IC50 200TP_TRANSPORTER: inhibition of Adefovir uptake in OAT1-expressing CHO cells [AID681160, Type: Literature]Solute carrier family 22 member 6 [gi:74762955]
View
12
[SID103179006]
Ki 488TP_TRANSPORTER: inhibition of PAH uptake in Xenopus laevis oocytes [AID681340, Type: Literature]Solute carrier family 22 member 6 [gi:81886651]
View
13
[SID103179006]
IC50 500Inhibition of human MATE1-mediated ASP+ uptake expressed in HEK293 cells after 1.5 mins by fluorescence assay [AID721754, Type: Literature]Multidrug and toxin extrusion protein 1 [gi:74731723]
View
14
[SID103179006]
DRUGMATRIX: Protein Serine/Threonine Kinase PKCalpha enzyme inhibition (substrate: Histone) [AID625179, Type: other]Protein kinase C alpha type [gi:317373571]
View
15
[SID103179006]
IC50 DRUGMATRIX: Serotonin (5-Hydroxytryptamine) 5-HT2C radioligand binding (ligand: [3H] Mesulergine) [AID625218, Type: confirmatory]5-hydroxytryptamine receptor 2C [gi:112816]
View
16
[SID103179006]
IC50 DRUGMATRIX: Carbonic Anhydrase II enzyme inhibition (substrate: 4-Nitrophenyl acetate (4-NPA)) [AID625236, Type: confirmatory]Carbonic anhydrase 2 [gi:115456]
View
17
[SID103179006]
IC50 DRUGMATRIX: Opiate mu (OP3, MOP) radioligand binding (ligand: [3H] Diprenorphine) [AID625163, Type: confirmatory]Mu-type opioid receptor [gi:2851402]
View
18
[SID103179006]
IC50 DRUGMATRIX: Serotonin (5-Hydroxytryptamine) 5-HT2B radioligand binding (ligand: [3H] Lysergic acid diethylamide) [AID625217, Type: confirmatory]5-hydroxytryptamine receptor 2B [gi:1168220]
View
19
[SID103179006]
Inhibition of human MATE1-mediated ASP+ uptake expressed in HEK293 cells at 20 uM after 1.5 mins by fluorescence assay [AID721753, Type: Literature]Multidrug and toxin extrusion protein 1 [gi:74731723]
View
20
[SID103179006]
IC50 DRUGMATRIX: Endothelin ETA radioligand binding (ligand: [125I] Endothelin-1) [AID625257, Type: confirmatory]Endothelin-1 receptor [gi:119606]
View