SureCN13211394 (CID 46882949) - BioAssay Data Summary for Compound
.
BioActivity Outcomes:
Active(7)
 
 
Unspecified(3)
 
 
Top Targets:
HAD like(3)
 
 
EHN(1)
 
 
BioAssay Types:
Literature(10)
 
 
 
BioActivity Types:
IC50(10)
 
 
 
SAR
Target summary
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 10    Data Row: 10   Total Pages: 1   
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#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID103743610]
IC50 0.001Inhibition of human soluble epoxide hydrolase [AID470609, Type: Literature]Bifunctional epoxide hydrolase 2 [gi:67476665]
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2
[SID103743610]
IC50 0.001Inhibition of human soluble epoxide hydrolase [AID470609, Type: Literature]Bifunctional epoxide hydrolase 2 [gi:67476665]
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3
[SID103743610]
IC50 0.015Inhibition of rat soluble epoxide hydrolase [AID470610, Type: Literature]Bifunctional epoxide hydrolase 2 [gi:462371]
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4
[SID103743610]
IC50 0.07Inhibition of potassium channel IKr [AID470617, Type: Literature]
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5
[SID103743610]
IC50 0.9Inhibition of potassium channel diltiazem binding site [AID470616, Type: Literature]
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6
[SID103743610]
IC50 1Inhibition of human soluble epoxide hydrolase in HEK293 cells assessed as DHET production [AID470611, Type: Literature]Bifunctional epoxide hydrolase 2 [gi:67476665]
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7
[SID103743610]
IC50 1Inhibition of human soluble epoxide hydrolase in HEK293 cells assessed as DHET production [AID470611, Type: Literature]Bifunctional epoxide hydrolase 2 [gi:67476665]
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8
[SID103743610]
IC50 10Inhibition of CYP2C9 [AID470613, Type: Literature]
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9
[SID103743610]
IC50 10Inhibition of CYP2D6 [AID470614, Type: Literature]
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10
[SID103743610]
IC50 10Inhibition of CYP3A4 [AID470615, Type: Literature]
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11
[SID103743610]
IC50 10Inhibition of Nav1.5 channel [AID470618, Type: Literature]
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12
[SID103743610]
IC50 100Inhibition of human microsomal epoxide hydrolase [AID470612, Type: Literature]Epoxide hydrolase 1 [gi:123926]
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