CHEMBL611600 (CID 46876435) - BioAssay Data Summary for Compound
.
BioActivity Outcomes:
Active(2)
 
 
Unspecified(5)
 
 
BioAssay Types:
Literature(7)
 
 
 
BioActivity Types:
Ki(2)
 
 
SAR
Target summary
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 7    Data Row: 7   Total Pages: 1   
Sort: [Click the result table header to sort]
#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID103732998]
Ki 0.05Binding affinity for adenosine A1 receptor in vitro using rat brain membranes. [AID32036, Type: Literature]
View
2
[SID103732998]
Ki 0.25Binding affinity for adenosine A2 receptor in vitro using rat striatal membrane. [AID33577, Type: Literature]
View
3
[SID103732998]
 Effective dose of compound for phenylbenzoquinone-Induced writhing in mice after peroral administration expressed as analgesic activity; Not dose dependent [AID131694, Type: Literature]
View
4
[SID103732998]
 Percent displacement from adenosine A1 receptor at 10e-5 M in rat brain membrane in vitro. [AID31255, Type: Literature]
View
5
[SID103732998]
 Percent displacement from adenosine A2 receptor at 10e-7 M in rat striatal membrane in vitro. [AID30813, Type: Literature]
View
6
[SID103732998]
 Percent displacement from adenosine A2 receptor at 10e-5 M in rat striatal membrane in vitro. [AID30812, Type: Literature]
View
7
[SID103732998]
 Percent displacement from adenosine A1 receptor at 10e-7 M in rat brain membrane in vitro. [AID31256, Type: Literature]
View