SureCN2903983 (CID 46868793) - BioAssay Data Summary for Compound
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BioActivity Outcomes:
Active(3)
 
 
Top Targets:
Orexin rec2(1)
 
 
BioAssay Types:
Literature(3)
 
 
BioActivity Types:
Ki(3)
 
 
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Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 3    Data Row: 3   Total Pages: 1   
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OutcomeTypeValue [μM]
1
[SID103755918]
Ki 0.0085Displacement of [3H](S)-N-(2-(1H-pyrrol-1-yl)phenyl)-1-(2-(1-methyl-1H-benzo[d]imidazol-2-ylthio)acetyl)pyrrolidine-2-carboxamide from human OX2R expressed in CHO cells after 3 hrs by scintillation counting [AID482635, Type: Literature]Orexin receptor type 2 [gi:206729885]
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2
[SID103755918]
Ki 0.0085Displacement of [3H](S)-N-(2-(1H-pyrrol-1-yl)phenyl)-1-(2-(1-methyl-1H-benzo[d]imidazol-2-ylthio)acetyl)pyrrolidine-2-carboxamide from human OX2R expressed in CHO cells after 3 hrs by scintillation counting [AID482635, Type: Literature]Orexin receptor type 2 [gi:206729885]
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3
[SID103755918]
Ki 0.054Displacement of [3H](S)-N-(biphenyl-2-yl)-1-(2-(1-methyl-1H-benzo[d]imidazol-2-ylthio)acetyl)pyrrolidine-2-carboxamide from human OX1R expressed in CHO cells after 3 hrs by scintillation counting [AID482633, Type: Literature]Orexin receptor type 1 [gi:205804177]
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4
[SID103755918]
Ki 0.054Displacement of [3H]N-cyclobutyl-5-methyl-N-(2-(1-methyl-1H-benzo[d]imidazol-2-ylthio)ethyl)-2-(2H-1,2,3-triazol-2-yl)benzamide from human OX1R expressed in CHO cells after 20 hrs by scintillation counting [AID482634, Type: Literature]Orexin receptor type 1 [gi:205804177]
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5
[SID103755918]
Ki 0.054Displacement of [3H](S)-N-(biphenyl-2-yl)-1-(2-(1-methyl-1H-benzo[d]imidazol-2-ylthio)acetyl)pyrrolidine-2-carboxamide from human OX1R expressed in CHO cells after 3 hrs by scintillation counting [AID482633, Type: Literature]Orexin receptor type 1 [gi:205804177]
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6
[SID103755918]
Ki 0.054Displacement of [3H]N-cyclobutyl-5-methyl-N-(2-(1-methyl-1H-benzo[d]imidazol-2-ylthio)ethyl)-2-(2H-1,2,3-triazol-2-yl)benzamide from human OX1R expressed in CHO cells after 20 hrs by scintillation counting [AID482634, Type: Literature]Orexin receptor type 1 [gi:205804177]
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