CHEMBL566041 (CID 45487435) - BioAssay Data Summary for Compound
.
BioActivity Outcomes:
Active(1)
 
 
Unspecified(1)
 
 
Top Targets:
7TM GPCR Srx(1)
 
 
BioAssay Types:
Literature(2)
 
 
 
BioActivity Types:
IC50(1)
 
 
SAR
Target summary
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Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 2    Data Row: 2   Total Pages: 1   
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#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID103707910]
IC50 0.00027Displacement of [125I]-PYY from human NPYY1 receptor overexpressed in CHO cell membrane after 120 mins by scintillation counting [AID447594, Type: Literature]Neuropeptide Y receptor type 1 [gi:128997]
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2
[SID103707910]
IC50 0.00027Displacement of [125I]-PYY from human NPYY1 receptor overexpressed in CHO cell membrane after 120 mins by scintillation counting [AID447594, Type: Literature]Neuropeptide Y receptor type 1 [gi:128997]
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3
[SID103707910]
 Octanol-water distribution coefficient log Dat pH 7.4 by water-plug aspiration/injection method combined with HPLC-mass spectrometry [AID447593, Type: Literature]
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