SR-03000001301 (CID 45100462) - BioAssay Data Summary for Compound
.
BioActivity Outcomes:
Active(1)
 
 
Inactive(2)
 
 
Top Targets:
Alpha TIF(1)
 
 
NR LBD Lrh-1(1)
 
 
NR LBD SF-1(1)
 
 
SAR
Target summary
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 3    Data Row: 3   Total Pages: 1   
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#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID92092824]
 Center Based Initiative to identify novel inverse agonists of the liver receptor homolog-1 (LRH1; NR5A2): Luminescence-based counterscreen assay to identify SF-1 inhibitors [AID488779, Type: other]steroidogenic factor-1 [Homo sapiens] [gi:216409744]
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2
[SID92092824]
 Center Based Initiative to identify novel inverse agonists of the liver receptor homolog-1 (LRH1; NR5A2): Luminescence-based counterscreen assay to identify SF-1 inhibitors [AID488779, Type: other]steroidogenic factor-1 [Homo sapiens] [gi:216409744]
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3
[SID92092824]
 Center Based Initiative to identify novel inverse agonists of the liver receptor homolog-1 (LRH1; NR5A2): Luminescence-based counterscreen assay to identify SF-1 inhibitors [AID488779, Type: other]steroidogenic factor-1 [Homo sapiens] [gi:216409744]
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4
[SID92092824]
 Center Based Initiative to identify novel inverse agonists of the liver receptor homolog-1 (LRH1; NR5A2): Luminescence-based counterscreen assay to identify inhibitors of the human herpes virus VP16 transcriptional activator protein (VP16) [AID488775, Type: other]transactivating tegument protein VP16 [Human herpesvirus 1] [gi:9629429]
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5
[SID92092824]
 Center Based Initiative to identify novel inverse agonists of the liver receptor homolog-1 (LRH-1; NR5A2): Luminescence-based primary assay to identify LRH1 inhibitors (3X%INH) [AID485348, Type: other]NR5A2 gene product [Homo sapiens] [gi:4504343]
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6
[SID92092824]
 Center Based Initiative to identify novel inverse agonists of the liver receptor homolog-1 (LRH-1; NR5A2): Luminescence-based primary assay to identify LRH1 inhibitors (3X%INH) [AID485348, Type: other]NR5A2 gene product [Homo sapiens] [gi:4504343]
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