CHEMBL473618 (CID 44572379) - BioAssay Data Summary for Compound
.
BioActivity Outcomes:
Active(3)
 
 
Unspecified(2)
 
 
BioAssay Types:
Literature(5)
 
 
 
SAR
Target summary
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 5    Data Row: 5   Total Pages: 1   
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#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID103611570]
 Antagonist activity at human luteinizing hormone receptor expressed in CHOK1 cells assessed as decrease in recombinant human chorionic gonadotropin activation potency at 10 uM by c-AMP-mediated luciferase assay [AID414566, Type: Literature]Lutropin-choriogonadotropic hormone receptor [gi:281185513]
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2
[SID103611570]
 Antagonist activity at human luteinizing hormone receptor expressed in CHOK1 cells assessed as decrease in recombinant human chorionic gonadotropin activation potency at 10 uM by c-AMP-mediated luciferase assay [AID414566, Type: Literature]Lutropin-choriogonadotropic hormone receptor [gi:281185513]
View
3
[SID103611570]
 Antagonist activity at human luteinizing hormone receptor expressed in CHOK1 cells assessed as decrease in recombinant human chorionic gonadotropin activation potency at 10 uM by c-AMP-mediated luciferase assay [AID414566, Type: Literature]Lutropin-choriogonadotropic hormone receptor [gi:281185513]
View
4
[SID103611570]
 Antagonist activity at human luteinizing hormone receptor expressed in CHOK1 cells assessed as decrease in Org 43553 activation potency at 10 uM by c-AMP-mediated luciferase assay [AID414567, Type: Literature]Lutropin-choriogonadotropic hormone receptor [gi:281185513]
View
5
[SID103611570]
 Antagonist activity at human luteinizing hormone receptor expressed in CHOK1 cells assessed as decrease in Org 43553 activation potency at 10 uM by c-AMP-mediated luciferase assay [AID414567, Type: Literature]Lutropin-choriogonadotropic hormone receptor [gi:281185513]
View
6
[SID103611570]
 Antagonist activity at human luteinizing hormone receptor expressed in CHOK1 cells assessed as decrease in Org 43553 activation potency at 10 uM by c-AMP-mediated luciferase assay [AID414567, Type: Literature]Lutropin-choriogonadotropic hormone receptor [gi:281185513]
View
7
[SID103611570]
 Antagonist activity at human luteinizing hormone receptor expressed in CHOK1 cells assessed as decrease in recombinant luteinizing hormone activation potency at 10 uM by c-AMP-mediated luciferase assay [AID414565, Type: Literature]Lutropin-choriogonadotropic hormone receptor [gi:281185513]
View
8
[SID103611570]
 Antagonist activity at human luteinizing hormone receptor expressed in CHOK1 cells assessed as decrease in recombinant luteinizing hormone activation potency at 10 uM by c-AMP-mediated luciferase assay [AID414565, Type: Literature]Lutropin-choriogonadotropic hormone receptor [gi:281185513]
View
9
[SID103611570]
 Antagonist activity at human luteinizing hormone receptor expressed in CHOK1 cells assessed as decrease in recombinant luteinizing hormone activation potency at 10 uM by c-AMP-mediated luciferase assay [AID414565, Type: Literature]Lutropin-choriogonadotropic hormone receptor [gi:281185513]
View
10
[SID103611570]
 Displacement of [3H]Org43553 from human luteinizing hormone receptor expressed in CHOK1 cells assessed as increase in radioligand dissociation at 10 uM by scintillation spectrometry relative to control [AID414561, Type: Literature]Lutropin-choriogonadotropic hormone receptor [gi:281185513]
View
11
[SID103611570]
 Displacement of [3H]Org43553 from human luteinizing hormone receptor expressed in CHOK1 cells assessed as increase in radioligand dissociation at 10 uM by scintillation spectrometry relative to control [AID414561, Type: Literature]Lutropin-choriogonadotropic hormone receptor [gi:281185513]
View
12
[SID103611570]
 Displacement of [3H]Org43553 from human luteinizing hormone receptor expressed in CHOK1 cells assessed as increase in radioligand dissociation at 10 uM by scintillation spectrometry relative to control [AID414561, Type: Literature]Lutropin-choriogonadotropic hormone receptor [gi:281185513]
View
13
[SID103611570]
 Displacement of [3H]Org43553 from human luteinizing hormone receptor expressed in CHOK1 cells at 10 uM by scintillation spectrometry [AID414560, Type: Literature]Lutropin-choriogonadotropic hormone receptor [gi:281185513]
View
14
[SID103611570]
 Displacement of [3H]Org43553 from human luteinizing hormone receptor expressed in CHOK1 cells at 10 uM by scintillation spectrometry [AID414560, Type: Literature]Lutropin-choriogonadotropic hormone receptor [gi:281185513]
View
15
[SID103611570]
 Displacement of [3H]Org43553 from human luteinizing hormone receptor expressed in CHOK1 cells at 10 uM by scintillation spectrometry [AID414560, Type: Literature]Lutropin-choriogonadotropic hormone receptor [gi:281185513]
View