Uridine Diphosphate N-Acetylglucosamine (CID 445675) - BioAssay Data Summary for Compound
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BioActivity Outcomes:
Active(4)
 
 
Inactive(1)
 
 
Unspecified(2)
 
 
Top Targets:
7TM GPCR Srx(1)
 
 
BioAssay Types:
Literature(7)
 
 
 
 
BioActivity Types:
EC50(2)
 
 
IC50(1)
 
 
SAR
Target summary
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 7    Data Row: 7   Total Pages: 1   
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#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID103516236]
Km 2The compound was tested for inhibition of the rate of 1 uM UDP-[3H]-GlcNAc import into the lumen of the Golgi membranes. [AID74260, Type: Literature]
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2
[SID103516236]
IC50 4Inhibitory concentration at which there is accumulation of UDP-[3H]-GlcNAc in the lumen of the Golgi membranes. [AID74253, Type: Literature]
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3
[SID103516236]
EC50 4.38Agonist activity at human P2Y14 expressed in COS7 cells assessed as stimulation of PLC-mediated [3H]inositol hydrolsis [AID286300, Type: Literature]
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4
[SID103516236]
EC50 4.38Agonist activity at human P2Y14 receptor expressed in human COS7 cells [AID450300, Type: Literature]P2Y purinoceptor 14 [gi:3122322]
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5
[SID103516236]
 Ratio of Vmax to Km for Neisseria meningitidis beta1,3-N-acetylglucosaminyltransferase LgtA assessed as enzyme catalyzed glycosylation using lactose as substrate after 2 to 30 mins by SAMDI analysis [AID613190, Type: Literature]Beta 1,3 N-acetylglucosaminyltransferase [gi:75448036]
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6
[SID103516236]
 Activity of Neisseria meningitidis beta1,3-N-acetylglucosaminyltransferase LgtA assessed as enzyme catalyzed glycosylation using lactose as substrate after 2 to 30 mins by SAMDI analysis [AID613189, Type: Literature]Beta 1,3 N-acetylglucosaminyltransferase [gi:75448036]
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7
[SID103516236]
 Agonist activity at human P2Y2 receptor expressed in human 1321N1 cells up to 10 uM [AID450303, Type: Literature]P2Y purinoceptor 2 [gi:311033490]
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