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Oleic Acid (CID 445639) - Compound BioActivity Data
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BioActivity Outcomes:
Active(51)
 
 
Inactive(1159)
 
 
Inconclusive(64)
 
 
Unspecified(108)
 
 
Top Targets:
7tm 4(39)
 
 
NR LBD PPAR(32)
 
 
 
 
NR LBD ER(25)
 
 
 
NR LBD AR(25)
 
 
 
NR LBD TR(19)
 
 
 
BioAssay Types:
Confirmatory(631)
 
 
 
 
 
Screening(406)
 
 
 
 
Literature(230)
 
 
 
 
 
Summary(63)
 
 
 
BioActivity Types:
Potency(526)
 
 
 
 
 
IC50(60)
 
 
 
 
 
Kd(10)
 
 
 
EC50(9)
 
 
 
Ki(6)
 
 
 
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 1015    Data Row: 1382   Total Pages: 70   Display: Page     
Sort: [Click the result table header to sort]
#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID46392022]
Kd 0.0085Experimentally measured binding affinity data (Kd) for protein-ligand complexes derived from PDB [AID977611, Type: Literature]Chain A, Human Serum Albumin Complexed With Cis-9-Octadecenoic Acid (Oleic Acid) [gi:18158774]
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2
[SID46392022]
Kd 0.0085Experimentally measured binding affinity data (Kd) for protein-ligand complexes derived from PDB [AID977611, Type: Literature]Chain A, Human Serum Albumin Complexed With Cis-9-Octadecenoic Acid (Oleic Acid) [gi:18158774]
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3
[SID46393429]
Kd 0.009Experimentally measured binding affinity data (Kd) for protein-ligand complexes derived from PDB [AID977611, Type: Literature]Chain A, Schistosoma Mansoni Fatty Acid Binding Protein In Complex With Oleic Acid [gi:55670477]
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4
[SID103167698]
Ki 0.18Displacement of 1-anilinonaphthalene-8-sulphonic acid from rat recombinant L-FABP high binding affinity site expressed in Escherichia coli BL21 by competitive fluorescence displacement assay [AID407366, Type: Literature]Fatty acid-binding protein, liver [gi:119810]
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5
[SID103167698]
Ki 0.185Displacement of 1,8-ANS from aFABP by fluorescence based-assay [AID307907, Type: Literature]
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6
[SID103167698]
Kd 0.2Binding affinity to L-FABP high binding affinity site by titration calorimetry method [AID407370, Type: Literature]
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7
[SID103167698]
Ki 0.248Displacement of 1,8-ANS from eFABP by fluorescence based-assay [AID307909, Type: Literature]
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8
[SID46391972]
Kd 0.3Experimentally measured binding affinity data (Kd) for protein-ligand complexes derived from PDB [AID977611, Type: Literature]Chain A, Toward Changing Specificity: Adipocyte Lipid Binding Protein Mutant, Oleic Acid Bound Form [gi:33356927]
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9
[SID46391972]
Kd 0.3Experimentally measured binding affinity data (Kd) for protein-ligand complexes derived from PDB [AID977611, Type: Literature]Chain A, Toward Changing Specificity: Adipocyte Lipid Binding Protein Mutant, Oleic Acid Bound Form [gi:33356927]
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10
[SID46392136]
Kd 0.43Experimentally measured binding affinity data (Kd) for protein-ligand complexes derived from PDB [AID977611, Type: Literature]Chain A, 1.4 Angstroms Structural Studies On Human Muscle Fatty Acid Binding Protein: Binding Interactions With Three Saturated And Unsaturated C18 Fatty Acids [gi:157831354]
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11
[SID46392136]
Kd 0.43Experimentally measured binding affinity data (Kd) for protein-ligand complexes derived from PDB [AID977611, Type: Literature]Chain A, 1.4 Angstroms Structural Studies On Human Muscle Fatty Acid Binding Protein: Binding Interactions With Three Saturated And Unsaturated C18 Fatty Acids [gi:157831354]
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12
[SID103167698]
IC50 0.6Inhibition of PPAR-alpha (unknown origin) by SPA assay [AID1094404, Type: confirmatory]Peroxisome proliferator-activated receptor alpha [gi:3041727]
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13
[SID103167698]
IC50 0.6Displacement of [3H]GW2331 from Homo sapiens (human) PPARalpha receptor by scintillation proximity assay [AID1114584, Type: confirmatory]Peroxisome proliferator-activated receptor alpha [gi:3041727]
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14
[SID103167698]
Kd 0.9Binding affinity to L-FABP low binding affinity site by titration calorimetry method [AID407371, Type: Literature]
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15
[SID103167698]
Ki 2.9Displacement of 1-anilinonaphthalene-8-sulphonic acid from rat recombinant L-FABP low binding affinity site expressed in Escherichia coli BL21 by competitive fluorescence displacement assay [AID407369, Type: Literature]Fatty acid-binding protein, liver [gi:119810]
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16
[SID103167698]
IC50 4.1Displacement of [3H]BRL49653 from Homo sapiens (human) PPARgamma receptor by scintillation proximity assay [AID1114583, Type: confirmatory]Peroxisome proliferator-activated receptor gamma [gi:13432234]
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17
[SID103167698]
IC50 5.3Displacement of [3H]GW2433 from Homo sapiens (human) PPARdelta receptor by scintillation proximity assay [AID1114582, Type: confirmatory]Peroxisome proliferator-activated receptor delta [gi:417522]
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18
[SID103167698]
GI50 10Growth inhibitory activity against human cancer cell line in the NCI's anticancer drug screening program [AID247402, Type: Literature]
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19
[SID26732603]
EC50 10.41Confirmation Dose Response screen for compounds that protect hERG from block by proarrhythmic agents [AID2121, Type: confirmatory]putative potassium channel subunit [Homo sapiens] [gi:487738]
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20
[SID26732603]
Potency 10.6213qHTS for Inhibitors of PLK1-PDB (polo-like kinase 1 - polo-box domain): Primary Screen [AID720504, Type: confirmatory]serine/threonine-protein kinase PLK1 [Homo sapiens] [gi:21359873]
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