CHEMBL461326
(CID
44562796
) -
BioAssay Data Summary for Compound
.
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BioActivity Outcomes:
Active(2)
BioAssay Types:
Literature(
2
)
BioActivity Types:
IC50(
1
)
Ki(
1
)
SAR
Target summary
Data download
Chemical Probe
Active
Inactive
Inconclusive
Unspecified
Total Bioassays: 2 Data Row: 2 Total Pages: 1
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#
Substance
Activity
BioAssay
Target
Links
Outcome
Type
Value [μM]
1
[SID
103588728
]
Active
Ki
0.2
Displacement of [33P]2-Mes-ADP from human recombinant P2Y1 receptor expressed in human U20S cells [AID
409975
, Type: Literature]
P2Y purinoceptor 1 [gi:
1352692
]
View
X
Row No.
1
Structure
Substance
SID
103588728
CID
44562796
Outcome
Active
Ki
0.2 [uM]
BioAssay
Displacement of [33P]2-Mes-ADP from human recombinant P2Y1 receptor expressed in human U20S cells
AID
409975
BioAssay type
Literature
Target
P2Y purinoceptor 1 [gi:
1352692
]
PubMed
18926700
Data Table
2
[SID
103588728
]
Active
IC50
0.8
Antagonist activity at human P2Y1 receptor in HEK293 cells assessed as intracellular calcium level by FLIPR [AID
409974
, Type: Literature]
P2Y purinoceptor 1 [gi:
1352692
]
View
X
Row No.
2
Structure
Substance
SID
103588728
CID
44562796
Outcome
Active
IC50
0.8 [uM]
BioAssay
Antagonist activity at human P2Y1 receptor in HEK293 cells assessed as intracellular calcium level by FLIPR
AID
409974
BioAssay type
Literature
Target
P2Y purinoceptor 1 [gi:
1352692
]
PubMed
18926700
Data Table
Chemical Probe 
Active 
Inactive 
Inconclusive 
Unspecified 
