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CHEMBL1162193 (CID 44457390) - Compound BioActivity Data
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BioActivity Outcomes:
Active(4)
 
 
Inactive(3)
 
 
Unspecified(1)
 
 
BioAssay Types:
Literature(8)
 
 
 
 
BioActivity Types:
EC50(5)
 
 
 
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 8    Data Row: 8   Total Pages: 1   
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#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID103762279]
EC50 0.2Agonist activity evaluated as change in the level of cytosolic calcium in 1321N astrocytoma cells infected with a retrovirus encoding the human P2Y6 receptor [AID89273, Type: Literature]
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2
[SID103762279]
EC50 0.4Agonist activity at P2Y6 receptor expressed in human 1321 cells by calcium mobilization assay [AID315757, Type: Literature]
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3
[SID103762279]
EC50 13.54Agonist activity at P2Y2 receptor expressed in human 1321 cells by calcium mobilization assay [AID315756, Type: Literature]
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4
[SID103762279]
EC50 22Agonist activity evaluated as change in the level of cytosolic calcium in 1321N astrocytoma cells infected with a retrovirus encoding the human P2Y2 receptor [AID89269, Type: Literature]
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5
[SID103762279]
EC50 100Agonist activity evaluated as change in the level of cytosolic calcium in 1321N astrocytoma cells infected with a retrovirus encoding the human P2Y4 receptor [AID89271, Type: Literature]
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6
[SID103762279]
Agonist activity at human recombinant P2Y1 receptor expressed in human 1321 cells at 100 uM by calcium mobilization assay [AID315758, Type: Literature]P2Y purinoceptor 1 [gi:1352692]
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7
[SID103762279]
Antagonist activity at P2Y12 receptor assessed as inhibition of ADP-induced human platelet aggregation by washed platelet assay at 100 uM [AID315754, Type: Literature]P2Y purinoceptor 12 [gi:21263835]
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8
[SID103762279]
Agonist activity evaluated as change in the level of cytosolic calcium in 1321N astrocytoma cells infected with a retrovirus encoding the human P2Y1 receptor at 100 uM; IA is inactive [AID89268, Type: Literature]
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