CHEMBL1162193 (CID 44457390) - BioAssay Data Summary for Compound
.
BioActivity Outcomes:
Active(2)
 
 
Inactive(2)
 
 
Top Targets:
7TM GPCR Srx(1)
 
 
BioAssay Types:
Literature(4)
 
 
 
BioActivity Types:
EC50(2)
 
 
SAR
Target summary
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 4    Data Row: 4   Total Pages: 1   
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#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID103762279]
EC50 0.4Agonist activity at P2Y6 receptor expressed in human 1321 cells by calcium mobilization assay [AID315757, Type: Literature]
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2
[SID103762279]
EC50 13.54Agonist activity at P2Y2 receptor expressed in human 1321 cells by calcium mobilization assay [AID315756, Type: Literature]
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3
[SID103762279]
 Agonist activity at human recombinant P2Y1 receptor expressed in human 1321 cells at 100 uM by calcium mobilization assay [AID315758, Type: Literature]P2Y purinoceptor 1 [gi:1352692]
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4
[SID103762279]
 Antagonist activity at P2Y12 receptor assessed as inhibition of ADP-induced human platelet aggregation by washed platelet assay at 100 uM [AID315754, Type: Literature]P2Y purinoceptor 12 [gi:21263835]
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