CHEMBL224873 (CID 44420924) - BioAssay Data Summary for Compound
.
BioActivity Outcomes:
Active(3)
 
 
Unspecified(2)
 
 
Top Targets:
7TM GPCR Srsx(4)
 
 
 
BioAssay Types:
Literature(5)
 
 
 
BioActivity Types:
Ki(3)
 
 
SAR
Target summary
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Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 5    Data Row: 5   Total Pages: 1   
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#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID103510836]
Ki 0.0736Displacement of [3H]CPPA from human adenosine A1 receptor expressed in CHO cells [AID281459, Type: Literature]Adenosine receptor A [gi:231473]
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2
[SID103510836]
Ki 0.0736Displacement of [3H]CPPA from human adenosine A1 receptor expressed in CHO cells [AID281459, Type: Literature]Adenosine receptor A [gi:231473]
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3
[SID103510836]
Ki 0.0736Displacement of [3H]CPPA from human adenosine A1 receptor expressed in CHO cells [AID281459, Type: Literature]Adenosine receptor A [gi:231473]
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4
[SID103510836]
Ki 0.09Displacement of [125I]I-AB-MECA from human adenosine A3 receptor expressed in CHO cells [AID281463, Type: Literature]Adenosine receptor A [gi:1351831]
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5
[SID103510836]
Ki 0.09Displacement of [125I]I-AB-MECA from human adenosine A3 receptor expressed in CHO cells [AID281463, Type: Literature]Adenosine receptor A [gi:1351831]
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6
[SID103510836]
Ki 0.277Displacement of [3H]CGS-21680 from human adenosine A2A receptor expressed in CHO cells [AID281461, Type: Literature]Adenosine receptor A2 [gi:543740]
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7
[SID103510836]
Ki 0.277Displacement of [3H]CGS-21680 from human adenosine A2A receptor expressed in CHO cells [AID281461, Type: Literature]Adenosine receptor A2 [gi:543740]
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8
[SID103510836]
Ki 0.277Displacement of [3H]CGS-21680 from human adenosine A2A receptor expressed in CHO cells [AID281461, Type: Literature]Adenosine receptor A2 [gi:543740]
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9
[SID103510836]
 Agonist activity at human adenosine A2B receptor expressed in CHO cells assessed as stimulation of cAMP production at 10 uM [AID281467, Type: Literature]Adenosine receptor A2 [gi:112938]
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10
[SID103510836]
 Maximum efficacy at human recombinant adenosine A3 receptor expressed in CHO cells assessed as inhibition of cAMP production at 10 uM relative to NECA [AID281469, Type: Literature]Adenosine receptor A [gi:1351831]
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11
[SID103510836]
 Maximum efficacy at human recombinant adenosine A3 receptor expressed in CHO cells assessed as inhibition of cAMP production at 10 uM relative to NECA [AID281469, Type: Literature]Adenosine receptor A [gi:1351831]
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