CHEMBL377463 (CID 44413583) - BioAssay Data Summary for Compound
.
BioActivity Outcomes:
Active(2)
 
 
Top Targets:
PTKc Abl(2)
 
 
BioAssay Types:
Literature(2)
 
 
BioActivity Types:
EC50(1)
 
 
IC50(1)
 
 
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 2    Data Row: 2   Total Pages: 1   
Sort: [Click the result table header to sort]
#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID103492918]
IC50 0.15Inhibition of c-ABL [AID266584, Type: Literature]Tyrosine-protein kinase ABL1 [gi:85681908]
View
2
[SID103492918]
IC50 0.15Inhibition of c-ABL [AID266584, Type: Literature]Tyrosine-protein kinase ABL1 [gi:85681908]
View
3
[SID103492918]
EC50 0.56Antiproliferative activity against K562 cells expressing Bcr-Abl [AID266585, Type: Literature]Tyrosine-protein kinase ABL1 [gi:85681908]
View
4
[SID103492918]
EC50 0.56Antiproliferative activity against K562 cells expressing Bcr-Abl [AID266585, Type: Literature]Tyrosine-protein kinase ABL1 [gi:85681908]
View