CHEMBL414719
(CID
44354499
) -
BioAssay Data Summary for Compound
.
BioActivity Outcomes:
Active(
3
)
Unspecified(2)
BioAssay Types:
Literature(
5
)
BioActivity Types:
Kd(
3
)
SAR
Target summary
Data download
Chemical Probe
Active
Inactive
Inconclusive
Unspecified
Total Bioassays: 5 Data Row: 5 Total Pages: 1
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#
Substance
Activity
BioAssay
Target
Links
Outcome
Type
Value [μM]
1
[SID
103368503
]
Active
Kd
0.00813
In vitro anti-oxytocic potency was recorded in absence of Mg2+ in rat uteri [AID
196972
, Type: Literature]
View
X
Row No.
1
Structure
Substance
SID
103368503
CID
44354499
Outcome
Active
Kd
0.00813 [uM]
BioAssay
In vitro anti-oxytocic potency was recorded in absence of Mg2+ in rat uteri
AID
196972
BioAssay type
Literature
Target
PubMed
7069719
Data Table
2
[SID
103368503
]
Active
Kd
0.01202
Compound evaluated in vivo and negative logarithm of effective dose divided by estimated volume of distribution (67 mL/kg) determined [AID
196817
, Type: Literature]
View
X
Row No.
2
Structure
Substance
SID
103368503
CID
44354499
Outcome
Active
Kd
0.01202 [uM]
BioAssay
Compound evaluated in vivo and negative logarithm of effective dose divided by estimated volume of distribution (67 mL/kg) determined
AID
196817
BioAssay type
Literature
Target
PubMed
7069719
Data Table
3
[SID
103368503
]
Active
Kd
0.01905
In vitro anti-oxytocic potency was recorded in presence of 0.5 mM Mg2+ in rat uteri [AID
196973
, Type: Literature]
View
X
Row No.
3
Structure
Substance
SID
103368503
CID
44354499
Outcome
Active
Kd
0.01905 [uM]
BioAssay
In vitro anti-oxytocic potency was recorded in presence of 0.5 mM Mg2+ in rat uteri
AID
196973
BioAssay type
Literature
Target
PubMed
7069719
Data Table
4
[SID
103368503
]
Unspecified
Effective dose for anti-vasopressor potency to reduce the response to 2x units of agonist to equal the response to 1x units [AID
179504
, Type: Literature]
View
X
Row No.
4
Structure
Substance
SID
103368503
CID
44354499
Outcome
Unspecified
BioAssay
Effective dose for anti-vasopressor potency to reduce the response to 2x units of agonist to equal the response to 1x units
AID
179504
BioAssay type
Literature
Target
PubMed
7069719
Data Table
5
[SID
103368503
]
Unspecified
Antidiuretic activity in intravenous antidiuretic assay in rats under ethanol anesthesia [AID
172980
, Type: Literature]
View
X
Row No.
5
Structure
Substance
SID
103368503
CID
44354499
Outcome
Unspecified
BioAssay
Antidiuretic activity in intravenous antidiuretic assay in rats under ethanol anesthesia
AID
172980
BioAssay type
Literature
Target
PubMed
7069719
Data Table