CHEMBL96273
(CID
44326476
) -
BioAssay Data Summary for Compound
.
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BioActivity Outcomes:
Active(3)
BioAssay Types:
Literature(
3
)
BioActivity Types:
Ki(
2
)
SAR
Target summary
Data download
Chemical Probe
Active
Inactive
Inconclusive
Unspecified
Total Bioassays: 3 Data Row: 3 Total Pages: 1
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#
Substance
Activity
BioAssay
Target
Links
Outcome
Type
Value [μM]
1
[SID
103305711
]
Active
Ki
0.00283
Binding affinity on HEK293 cells transiently transfected with plasmids encoding the rat Opioid receptor kappa 1 [AID
148568
, Type: Literature]
View
X
Row No.
1
Structure
Substance
SID
103305711
CID
44326476
Outcome
Active
Ki
0.00283 [uM]
BioAssay
Binding affinity on HEK293 cells transiently transfected with plasmids encoding the rat Opioid receptor kappa 1
AID
148568
BioAssay type
Literature
Target
PubMed
10893314
Data Table
2
[SID
103305711
]
Active
Ki
0.876
Binding affinity on HEK293 cells transiently transfected with plasmids encoding the rat Opioid receptor mu 1 [AID
151614
, Type: Literature]
View
X
Row No.
2
Structure
Substance
SID
103305711
CID
44326476
Outcome
Active
Ki
0.876 [uM]
BioAssay
Binding affinity on HEK293 cells transiently transfected with plasmids encoding the rat Opioid receptor mu 1
AID
151614
BioAssay type
Literature
Target
PubMed
10893314
Data Table
3
[SID
103305711
]
Active
Opioid receptor kappa 1 Antagonism (100 nM) is expressed as (Ke = [antagonist] / (IC50 ratio -1) [AID
148975
, Type: Literature]
View
X
Row No.
3
Structure
Substance
SID
103305711
CID
44326476
Outcome
Active
BioAssay
Opioid receptor kappa 1 Antagonism (100 nM) is expressed as (Ke = [antagonist] / (IC50 ratio -1)
AID
148975
BioAssay type
Literature
Target
PubMed
10893314
Data Table