CHEMBL96273 (CID 44326476) - BioAssay Data Summary for Compound
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BioActivity Outcomes:
Active(3)
 
 
BioAssay Types:
Literature(3)
 
 
BioActivity Types:
Ki(2)
 
 
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Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 3    Data Row: 3   Total Pages: 1   
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#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID103305711]
Ki 0.00283Binding affinity on HEK293 cells transiently transfected with plasmids encoding the rat Opioid receptor kappa 1 [AID148568, Type: Literature]
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2
[SID103305711]
Ki 0.876Binding affinity on HEK293 cells transiently transfected with plasmids encoding the rat Opioid receptor mu 1 [AID151614, Type: Literature]
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3
[SID103305711]
Opioid receptor kappa 1 Antagonism (100 nM) is expressed as (Ke = [antagonist] / (IC50 ratio -1) [AID148975, Type: Literature]
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