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Staurosporine (CID 44299148) - Compound BioActivity Data
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BioActivity Outcomes:
Active(1373)
 
 
Inactive(25)
 
 
Inconclusive(34)
 
 
Unspecified(748)
 
 
Top Targets:
PTKc Abl(39)
 
 
 
CYCLIN(38)
 
 
 
PTKc EGFR(31)
 
 
 
PTKc EphR A(25)
 
 
 
STKc RSK N(24)
 
 
 
BioAssay Types:
Literature(2142)
 
 
 
 
 
Confirmatory(37)
 
 
BioActivity Types:
Kd(885)
 
 
 
 
IC50(549)
 
 
 
 
 
EC50(15)
 
 
 
Ki(10)
 
 
 
 
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 2033    Data Row: 2180   Total Pages: 109   Display: Page     
Sort: [Click the result table header to sort]
#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID103243222]
IC50 4e-06Cytotoxicity against human HeLa cells after 48 hrs by MTT assay [AID595221, Type: Literature]
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2
[SID103243222]
IC50 4e-06Cytotoxicity against human HeLa cells after 48 hrs by MTT assay [AID600820, Type: Literature]
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3
[SID103243222]
Kd 2e-05Average Binding Constant for SLK; NA=Not Active at 10 uM [AID256578, Type: Literature]STE20-like serine/threonine-protein kinase [gi:74762732]
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4
[SID103243222]
Kd 2.4e-05Binding constant for SLK kinase domain [AID625086, Type: Literature]STE20-like serine/threonine-protein kinase [gi:74762732]
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5
[SID103243222]
Kd 2.4e-05Binding constant for SLK kinase domain [AID435832, Type: Literature]STE20-like serine/threonine-protein kinase [gi:74762732]
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6
[SID103243222]
Kd 3e-05Average Binding Constant for STK10; NA=Not Active at 10 uM [AID256604, Type: Literature]Serine/threonine-protein kinase 10 [gi:12643358]
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7
[SID103243222]
Kd 3.7e-05Binding constant for LOK kinase domain [AID435677, Type: Literature]Serine/threonine-protein kinase 10 [gi:12643358]
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8
[SID103243222]
Kd 3.7e-05Binding constant for LOK kinase domain [AID625030, Type: Literature]Serine/threonine-protein kinase 10 [gi:12643358]
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9
[SID103243222]
Kd 3.9e-05Binding constant for CAMKK1 kinase domain [AID435521, Type: Literature]Calcium/calmodulin-dependent protein kinase kinase 1 [gi:56404620]
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10
[SID103243222]
Kd 3.9e-05Binding constant for CAMKK1 kinase domain [AID625143, Type: Literature]Calcium/calmodulin-dependent protein kinase kinase 1 [gi:56404620]
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11
[SID103243222]
Kd 5e-05Average Binding Constant for CAMKK1; NA=Not Active at 10 uM [AID256583, Type: Literature]Calcium/calmodulin-dependent protein kinase kinase 1 [gi:56404620]
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12
[SID103243222]
Kd 5e-05Average Binding Constant for CAMKK2; NA=Not Active at 10 uM [AID256580, Type: Literature]Calcium/calmodulin-dependent protein kinase kinase 2 [gi:317373374]
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13
[SID103243222]
IC50 7e-05Inhibition of ROS1 by HotSpot assay relative to control [AID429341, Type: Literature]
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14
[SID103243222]
IC50 8e-05Inhibition Protein kinase C (PKC) [AID165147, Type: Literature]
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15
[SID103243222]
Kd 8.6e-05Binding constant for SNARK kinase domain [AID625139, Type: Literature]NUAK family SNF1-like kinase 2 [gi:74761376]
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16
[SID103243222]
Kd 8.6e-05Binding constant for SNARK kinase domain [AID435559, Type: Literature]NUAK family SNF1-like kinase 2 [gi:74761376]
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17
[SID103243222]
IC50 0.0001Inhibition of CAMK2B [AID350254, Type: Literature]
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18
[SID103243222]
IC50 0.0001Inhibition of CHK1 [AID350257, Type: Literature]
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19
[SID103243222]
IC50 0.0001Inhibition of PDGFRalpha [AID350286, Type: Literature]
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20
[SID103243222]
IC50 0.0001Inhibition of PHKgamma2 [AID350287, Type: Literature]
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