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CHEMBL51204 (CID 44295810) - Compound BioActivity Data
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BioActivity Outcomes:
Active(7)
 
 
Unspecified(4)
 
 
Top Targets:
7tm 4(2)
 
 
BioAssay Types:
Literature(11)
 
 
 
BioActivity Types:
Ki(9)
 
 
 
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 11    Data Row: 11   Total Pages: 1   
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#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID103235344]
Ki 6e-06Antagonist activity on agonist (U50,488) stimulated [35S]GTP-gamma-S, binding in cloned opioid receptor kappa 1 [AID147989, Type: Literature]
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2
[SID103235344]
Ki 2e-05Inhibition of stimulation of [35S]GTP-gamma-S, binding produced by the selective agonist (U69593, kappa-receptor), in guinea pig caudate membranes. [AID149438, Type: Literature]Kappa-type opioid receptor [gi:730228]
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3
[SID103235344]
Ki 0.00032Binding affinity to opioid receptor kappa 1 of guinea pig brain, using [3H]U-69593 as radioligand [AID149269, Type: Literature]Kappa-type opioid receptor [gi:730228]
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4
[SID103235344]
Ki 0.00216Inhibition of stimulation of [35S]GTP-gamma-S, binding produced by the selective agonist (DAMGO, mu-receptor), in guinea pig caudate membranes. [AID152228, Type: Literature]Mu-type opioid receptor [gi:3024265]
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5
[SID103235344]
Ki 0.00342Antagonist activity on agonist (DAMGO) stimulated [35S]GTP-gamma-S, binding in cloned mu opioid receptors. [AID152378, Type: Literature]
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6
[SID103235344]
Ki 0.00373Binding affinity to mu-opioid receptor of rat brain using [3H]DAMGO as radioligand. [AID152382, Type: Literature]
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7
[SID103235344]
Ki 0.301Binding affinity to delta-opioid receptor of rat brain using [3H]DADLE as radioligand. [AID149789, Type: Literature]
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8
[SID103235344]
Ki 0.1Antagonist activity on agonist (SNC-80) stimulated [35S]GTP-gamma-S, binding in cloned opioid receptor mu1 [AID152234, Type: Literature]
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9
[SID103235344]
Ki 0.3Inhibition of stimulation of [35S]GTP-gamma-S, binding produced by the selective agonist (SNC-80, delta-receptor), in guinea pig caudate membranes [AID150035, Type: Literature]
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10
[SID103235344]
delta/kappa ratio of the compound. [AID234390, Type: Literature]
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11
[SID103235344]
mu/kappa ratio of the compound. [AID234392, Type: Literature]
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