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CHEMBL414508 (CID 44283513) - Compound BioActivity Data
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BioActivity Outcomes:
Active(2)
 
 
Unspecified(5)
 
 
BioAssay Types:
Literature(7)
 
 
 
BioActivity Types:
Ki(3)
 
 
 
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 7    Data Row: 7   Total Pages: 1   
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#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID103210857]
Ki 0.0036In vitro antagonist activity was measured by inhibition of vasopressin-stimulated adenylate cyclase in renal medullary preparation in pig [AID217543, Type: Literature]Vasopressin V2 receptor [gi:418172]
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2
[SID103210857]
In vitro antagonist activity was measured by inhibition of binding of [3H]LVP to renal medullary membrane preparation in pig [AID159553, Type: Literature]
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3
[SID103210857]
Ki 1100In vitro antagonist activity was measured by inhibition of vasopressin-stimulated adenylate cyclase in renal medullary preparation in dog [AID217365, Type: Literature]
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4
[SID103210857]
Ki 3600In vitro antagonist activity was measured by inhibition of vasopressin-stimulated adenylate cyclase in renal medullary preparation in human [AID217522, Type: Literature]
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5
[SID103210857]
In vitro antagonist activity was measured by dose required to lower urine osmolality to 300 mOsm/kg of H2O [AID177219, Type: Literature]
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6
[SID103210857]
Antagonist activity was measured by maximum urine osmolality with a dose of 100 ug/kg peptide after pretreatment with indomethacin in dog [AID62810, Type: Literature]
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7
[SID103210857]
Antagonist activity was measured by maximum urine flow with a dose of 100 ug/kg peptide [AID63427, Type: Literature]
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