SureCN8558469 (CID 44279376) - BioAssay Data Summary for Compound
.
BioActivity Outcomes:
Active(3)
 
 
Inconclusive(2)
 
 
Unspecified(1)
 
 
Top Targets:
PTKc HER2(2)
 
 
Firefly Luc l..(1)
 
 
BioAssay Types:
Literature(3)
 
 
 
Confirmatory(3)
 
 
 
BioActivity Types:
Potency(3)
 
 
 
IC50(2)
 
 
SAR
Target summary
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 6    Data Row: 6   Total Pages: 1   
Sort: [Click the result table header to sort]
#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID103203166]
IC50 0.56Inhibition of rat Receptor protein-tyrosine kinase erbB2 [AID197676, Type: Literature]Receptor tyrosine-protein kinase erbB-2 [gi:3915663]
View
2
[SID103203166]
IC50 1.3Inhibition of c-erbB-2 overexpressing HB4a cell proliferation [AID79614, Type: Literature]Receptor tyrosine-protein kinase erbB-2 [gi:119533]
View
3
[SID103203166]
IC50 1.3Inhibition of c-erbB-2 overexpressing HB4a cell proliferation [AID79614, Type: Literature]Receptor tyrosine-protein kinase erbB-2 [gi:119533]
View
4
[SID124349913]
Potency 16.3432qHTS Assay for Inhibitors of Firefly Luciferase from the GSK Published Protein Kinase Inhibitor Set [AID652016, Type: confirmatory]Luciferase [Photinus pyralis] [gi:160794]
View
5
[SID103203166]
 Selectivity for EGF receptor and c-erbB-2 [AID235148, Type: Literature]
View
6
[SID124349913]
Potency 18.3374qHTS Assay for Inhibitors of Sea Pansy Luciferase from the GSK Published Protein Kinase Inhibitor Set [AID652015, Type: confirmatory]Renilla-luciferin 2-monooxygenase (EC 1.13.12.5) - sea pansy (Renilla reniformis) (fragment) [gi:84399]
View
7
[SID124349913]
Potency 25.0176qHTS for Inhibitors of binding or entry into cells for Lassa Virus [AID540256, Type: confirmatory]
View