BRD-K58130477-001-01-3
(CID
43816465
) -
BioAssay Data Summary for Compound
.
BioActivity Outcomes:
Active(
1
)
Inactive(
2
)
Top Targets:
CD36(
2
)
BioAssay Types:
Confirmatory(
3
)
BioActivity Types:
AC50(
3
)
SAR
Target summary
Data download
Chemical Probe
Active
Inactive
Inconclusive
Unspecified
Total Bioassays: 3 Data Row: 3 Total Pages: 1
Sort:
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#
Substance
Activity
BioAssay
Target
Links
Outcome
Type
Value [μM]
1
[SID
125082042
]
Active
AC50
0.386
HTS using DiI-HDL to assay lipid transfer in ldlA[SR-BI] cells Measured in Cell-Based System Using Plate Reader - 2085-01_Inhibitor_Dose_DryPowder_Activity_Set2 [AID
588392
, Type: confirmatory]
Scarb1 gene product [Mus musculus] [gi:
14389423
]
View
X
Row No.
1
Structure
Substance
SID
125082042
CID
43816465
Outcome
Active
AC50
0.386 [uM]
BioAssay
HTS using DiI-HDL to assay lipid transfer in ldlA[SR-BI] cells Measured in Cell-Based System Using Plate Reader - 2085-01_Inhibitor_Dose_DryPowder_Activity_Set2
AID
588392
BioAssay type
confirmatory
Target
Scarb1 gene product [Mus musculus] [gi:
14389423
]
PubMed
Data Table
2
[SID
125082042
]
Inactive
AC50
70
HDL Counter Assay: 3/24 Cytotox Measured in Cell-Based System Using Plate Reader - 2085-02_Inhibitor_Dose_DryPowder_Activity_Set5 [AID
602126
, Type: confirmatory]
View
X
Row No.
2
Structure
Substance
SID
125082042
CID
43816465
Outcome
Inactive
AC50
70 [uM]
BioAssay
HDL Counter Assay: 3/24 Cytotox Measured in Cell-Based System Using Plate Reader - 2085-02_Inhibitor_Dose_DryPowder_Activity_Set5
AID
602126
BioAssay type
confirmatory
Target
PubMed
Data Table
3
[SID
125082042
]
Inactive
AC50
DiI Quencher Assay Measured in Biochemical System Using Plate Reader - 2085-08_Inhibitor_Dose_DryPowder_Activity [AID
588403
, Type: confirmatory]
Scarb1 gene product [Mus musculus] [gi:
14389423
]
View
X
Row No.
3
Structure
Substance
SID
125082042
CID
43816465
Outcome
Inactive
AC50
[uM]
BioAssay
DiI Quencher Assay Measured in Biochemical System Using Plate Reader - 2085-08_Inhibitor_Dose_DryPowder_Activity
AID
588403
BioAssay type
confirmatory
Target
Scarb1 gene product [Mus musculus] [gi:
14389423
]
PubMed
Data Table