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DEET (CID 4284) - Compound BioActivity Data
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BioActivity Outcomes:
Active(11)
 
 
Inactive(1034)
 
 
Inconclusive(62)
 
 
Unspecified(20)
 
 
Top Targets:
NR LBD PPAR(34)
 
 
 
NR LBD ER(25)
 
 
 
NR LBD AR(25)
 
 
 
7TM GPCR Srx(19)
 
 
NR LBD TR(19)
 
 
 
BioAssay Types:
Confirmatory(546)
 
 
 
 
 
Screening(351)
 
 
 
Literature(84)
 
 
 
 
 
Summary(72)
 
 
 
 
BioActivity Types:
Potency(549)
 
 
 
 
 
IC50(11)
 
 
Kd(4)
 
 
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 753    Data Row: 1127   Total Pages: 57   Display: Page     
Sort: [Click the result table header to sort]
#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID144204654]
Potency-Replicate_1 2.6603qHTS assay to identify small molecule agonists of the estrogen receptor alpha (ER-alpha) signaling pathway using the BG1 cell line [AID743079, Type: confirmatory]estrogen nuclear receptor alpha [Homo sapiens] [gi:348019627]
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2
[SID144204654]
Potency-Replicate_1 21.3138qHTS assay to identify small molecule agonists of the estrogen receptor alpha (ER-alpha) signaling pathway [AID743075, Type: confirmatory]estrogen nuclear receptor alpha [Homo sapiens] [gi:348019627]
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3
[SID26747323]
Potency 25.1189qHTS Assay for Inhibitors of HPGD (15-Hydroxyprostaglandin Dehydrogenase) [AID894, Type: confirmatory]15-hydroxyprostaglandin dehydrogenase [NAD(+)] isoform 1 [Homo sapiens] [gi:31542939]
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4
[SID144204654]
Ratio Potency (uM) 25.797qHTS assay to identify small molecule agonists of the estrogen receptor alpha (ER-alpha) signaling pathway: Summary [AID743077, Type: summary]estrogen nuclear receptor alpha [Homo sapiens] [gi:348019627]
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5
[SID170483384]
Kd 31.3Experimentally measured binding affinity data (Kd) for protein-ligand complexes derived from PDB [AID977611, Type: Literature]Chain A, Crystal Structure Of Odorant Binding Protein 1 From Anopheles Gambiae (Agamobp1) With Deet (N,N-Diethyl-Meta-Toluamide) And Peg [gi:335892259]
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6
[SID170483384]
Kd 31.3Experimentally measured binding affinity data (Kd) for protein-ligand complexes derived from PDB [AID977611, Type: Literature]Chain A, Crystal Structure Of Odorant Binding Protein 1 From Anopheles Gambiae (Agamobp1) With Deet (N,N-Diethyl-Meta-Toluamide) And Peg [gi:335892259]
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7
[SID170483384]
Kd 31.3Experimentally measured binding affinity data (Kd) for protein-ligand complexes derived from PDB [AID977611, Type: Literature]Chain B, Crystal Structure Of Odorant Binding Protein 1 From Anopheles Gambiae (Agamobp1) With Deet (N,N-Diethyl-Meta-Toluamide) And Peg [gi:335892260]
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8
[SID170483384]
Kd 31.3Experimentally measured binding affinity data (Kd) for protein-ligand complexes derived from PDB [AID977611, Type: Literature]Chain B, Crystal Structure Of Odorant Binding Protein 1 From Anopheles Gambiae (Agamobp1) With Deet (N,N-Diethyl-Meta-Toluamide) And Peg [gi:335892260]
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9
[SID144209178]
Potency-Replicate_1 60.5094qHTS assay to identify small molecule that activate the aryl hydrocarbon receptor (AhR) signaling pathway [AID743085, Type: confirmatory]aryl hydrocarbon receptor [Homo sapiens] [gi:51095037]
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10
[SID48415187]
DSSTox (EPAFHM) EPA Fathead Minnow Acute Toxicity [AID1188, Type: other]
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11
[SID56320635]
Aqueous Solubility from MLSMR Stock Solutions [AID1996, Type: other]
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12
[SID8150108]
Screen for compounds that selectively inhibit cytochrome c release from purified mitochondria (CytoCRel) [AID1603, Type: other]
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13
[SID8150108]
Screen for compounds that inhibit polyglutamine induced protein aggregation (AGREG) [AID1604, Type: other]
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14
[SID8150108]
Screening of compounds showing protective effect against cell death induced by familial amyotrophic lateral sclerosis (FALS)-linked mutantsuperoxide dismutase 1 (SOD1) (ALSOD1) [AID1605, Type: other]
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15
[SID26747323]
qHTS profiling for inhibitors of Plasmodium falciparum proliferation [AID504749, Type: Literature]
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16
[SID124958332]
Inhibition of sodium fluorescein uptake in OATP1B1-transfected CHO cells at an equimolar substrate-inhibitor concentration of 10 uM [AID977599, Type: Literature]
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17
[SID124958332]
Inhibition of sodium fluorescein uptake in OATP1B3-transfected CHO cells at an equimolar substrate-inhibitor concentration of 10 uM [AID977602, Type: Literature]
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18
[SID8150108]
Assay to identify inhibitors of polyglutamine-induced caspase-3 activation (CASP3) [AID1583, Type: other]
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19
[SID8150108]
Yeast cell-based screen for compounds that suppress polyglutamine aggregation in vivo (75Q-TubU) [AID1593, Type: other]
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20
[SID8150108]
Screen for compounds that correct neuronal dysfunction without cell death as induced by the expression of polyglutamine-expanded, N-terminal huntingtin in C. elegans mechanosensory neurons (HDELENEU) [AID1599, Type: other]
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