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SID7969543 (CID 4076092) - Compound BioActivity Data
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BioActivity Outcomes:
Probe(1)
 
 
Active(11)
 
 
Inactive(915)
 
 
Inconclusive(20)
 
 
Unspecified(9)
 
 
Top Targets:
7tm 4(53)
 
 
alkPPc(14)
 
 
Tryp SPc(13)
 
 
Bcl-2 like(12)
 
 
Pyr redox dim(9)
 
 
BioAssay Types:
Screening(581)
 
 
 
 
 
Confirmatory(327)
 
 
 
 
 
Literature(20)
 
 
 
 
Summary(1)
 
 
BioActivity Types:
Potency(253)
 
 
 
 
IC50(50)
 
 
 
 
EC50(11)
 
 
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 859    Data Row: 956   Total Pages: 48   Display: Page     
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#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID7969543]
Summary of probe development efforts to identify inhibitors of the nuclear receptor Steroidogenic Factor 1 (SF-1). [AID1844, Type: summary]steroidogenic factor-1 [Homo sapiens] [gi:216409744]
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2
[SID103565235]
IC50 0.76Inhibition of GAL4-tagged NR5A1 by luciferase assay [AID329653, Type: Literature]
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3
[SID56436610]
Parallel artificial membrane permeability assay at pH 7.4 [AID624339, Type: other]
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4
[SID7969543]
Cell signaling CRE-BLA (Fsk stim) [AID662, Type: confirmatory]
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5
[SID7969543]
HTS of Estrogen Receptor- alpha Coactivator Binding Potentiators [AID639, Type: screening]Estrogen receptor 1 [Homo sapiens] [gi:118764400]
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6
[SID7969543]
Luminescence-based cell-based high throughput confirmation assay for inverse agonists of the liver receptor homolog-1 (LRH-1; NR5A2) [AID651613, Type: screening]nuclear receptor subfamily 5 group A member 2 isoform 2 [Homo sapiens] [gi:4504343]
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7
[SID7969543]
Primary biochemical high-throughput screening assay to measure P97 ATPase inhibition [AID1481, Type: screening]Valosin-containing protein [Homo sapiens] [gi:111305821]
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8
[SID7969543]
Counterscreen for inverse agonists of the liver receptor homolog-1 (LRH-1; NR5A2): Luminescence-based cell-based high throughput assay to identify inverse agonists of the Steroidogenic Factor 1 Nuclear Receptor (SF1; NR5A1) [AID651614, Type: screening]steroidogenic factor 1 [Homo sapiens] [gi:20070193]
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9
[SID7969543]
Dose-response cell-based assay for inhibitors of the nuclear receptor Steroidogenic Factor 1 (SF-1) [AID600, Type: confirmatory]steroidogenic factor 1 [Homo sapiens] [gi:20070193]
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10
[SID7969543]
Primary Cell-based High Throughput Screening assay for inhibitors of the nuclear receptor Steroidogenic Factor 1 (SF-1) [AID525, Type: screening]steroidogenic factor 1 [Homo sapiens] [gi:20070193]
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11
[SID56436610]
Inhibition of the MLL-AF4-AF9 Interaction in Pediatric Leukemia Measured in Biochemical System Using Plate Reader - 2160-01_Inhibitor_SinglePoint_HTS_Activity [AID651704, Type: screening]protein AF-9 isoform a [Homo sapiens] [gi:156104889]
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12
[SID7969543]
Luminescence-based cell-based primary high throughput screening assay to identify activators of the GAA850 frataxin (FXN) promoter [AID540364, Type: screening] [geneid:2395]
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13
[SID103565235]
IC50 33Inhibition of GAL4-tagged RORalpha by luciferase assay [AID329655, Type: Literature]
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14
[SID103565235]
IC50 33Inhibition of HSV1 GAL4-tagged VP16 by luciferase assay [AID329657, Type: Literature]
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15
[SID56436610]
Plasma Stability Mouse - Set 2 [AID624419, Type: other]
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16
[SID56436610]
Plasma Stability Human - 2 [AID624420, Type: other]
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17
[SID56436610]
Mouse hepatic microsome stability - Set 2 [AID624451, Type: screening]
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18
[SID56436610]
Human hepatic microsome stability-Set 2 [AID624452, Type: screening]
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19
[SID56436610]
Early assessment of compound stability in 1x PBS - Set 2 [AID624456, Type: other]
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20
[SID7969543]
Assay for HTS of Gi/Go-linked GPCRs using mGluR8: Primary Screening [AID488969, Type: screening]metabotropic glutamate receptor 8 [Rattus norvegicus] [gi:1575471]
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