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Meclofenoxate (CID 4039) - Compound BioActivity Data
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BioActivity Outcomes:
Active(3)
 
 
Inactive(312)
 
 
Inconclusive(35)
 
 
Unspecified(11)
 
 
Top Targets:
p450(18)
 
 
 
 
HSD10-like SD..(8)
 
 
7TM GPCR Srx(6)
 
 
P53(5)
 
 
PLN02808(5)
 
 
BioAssay Types:
Confirmatory(242)
 
 
 
 
Literature(73)
 
 
 
 
Screening(18)
 
 
BioActivity Types:
Potency(195)
 
 
 
IC50(2)
 
 
 
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 210    Data Row: 361   Total Pages: 19   Display: Page     
Sort: [Click the result table header to sort]
#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID11111000]
p450-cyp1a2 [AID410, Type: confirmatory]cytochrome P450 1A2 [Homo sapiens] [gi:73915100]
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2
[SID11110999]
p450-cyp1a2 [AID410, Type: confirmatory]cytochrome P450 1A2 [Homo sapiens] [gi:73915100]
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3
[SID11111000]
Cytochrome panel assay with activity outcomes [AID1851_4, Type: other]cytochrome P450 1A2 [Homo sapiens] [gi:73915100]
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4
[SID103252134]
IC50 500Inhibitory activity against Plasmodium falciparum [AID158688, Type: Literature]
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5
[SID103252134]
Literature-mined compound from Fourches et al multi-species drug-induced liver injury (DILI) dataset, effect in humans [AID588211, Type: Literature]
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6
[SID103252134]
Literature-mined compound from Fourches et al multi-species drug-induced liver injury (DILI) dataset, effect in rodents [AID588212, Type: Literature]
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7
[SID103252134]
Literature-mined compound from Fourches et al multi-species drug-induced liver injury (DILI) dataset, effect in non-rodents [AID588213, Type: Literature]
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8
[SID11110999]
Cytochrome panel assay with activity outcomes [AID1851, Type: other]
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9
[SID11111000]
qHTS profiling for inhibitors of Plasmodium falciparum proliferation [AID504749, Type: Literature]
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10
[SID11111000]
Cytochrome panel assay with activity outcomes [AID1851, Type: other]
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11
[SID103252134]
Time of recovery of righting reflux (RRT) in seconds was measured after administration of 200 mg/kg perorally in mice for the promotional effect on recovery from coma [AID119185, Type: Literature]
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12
[SID103252134]
Time of recovery of spontaneous movement (SMT) in seconds was measured after administration of 200 mg/kg perorally in mice for the promotional effect on recovery from coma [AID119402, Type: Literature]
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13
[SID103252134]
Antihypoxic effect tested by the survival time (SVT) in mice at a dose of 100 mg/kg [AID119554, Type: Literature]
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14
[SID103252134]
Antihypoxic effect by the survival time (SVT) in mice at a dose of 3 mg/kg administered intravenously in mice [AID119565, Type: Literature]
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15
[SID11111000]
Potency 0.2818qHTS Assay for Inhibitors of GCN5L2 [AID504327, Type: confirmatory]histone acetyltransferase KAT2A [Homo sapiens] [gi:153791535]
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16
[SID11111000]
Potency 0.5725Primary qHTS for delayed death inhibitors of the malarial parasite plastid, 48 hour incubation [AID504832, Type: confirmatory]
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17
[SID11111000]
Potency 0.9762S16 Schwann cell PMP22 intronic element firefly luciferase assay [AID624032, Type: confirmatory]peripheral myelin protein 22 [Rattus norvegicus] [gi:8393992]
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18
[SID11110999]
Potency 1.2589qHTS Assay for Activators of Cytochrome P450 3A4 [AID885, Type: confirmatory]cytochrome P450 3A4 isoform 1 [Homo sapiens] [gi:13435386]
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19
[SID11111000]
Potency 2.5575Primary qHTS for delayed death inhibitors of the malarial parasite plastid, 96 hour incubation [AID504834, Type: confirmatory]
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20
[SID90341454]
Potency 8.4921qHTS screen for enhancers of Arylsulfatase A (ASA1): LOPAC Validation Assay [AID720538, Type: confirmatory]arylsulfatase A [Homo sapiens] [gi:220983390]
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