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adinazolam (CID 37632) - Compound BioActivity Data
.
BioActivity Outcomes:
Unspecified(36)
 
 
Top Targets:
p450(1)
 
 
BioAssay Types:
Literature(36)
 
 
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 36    Data Row: 36   Total Pages: 1   
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#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID103304585]
log (1/Km) value for human liver microsome cytochrome P450 3A4 [AID243422, Type: Literature]Cytochrome P450 3A4 [gi:116241312]
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2
[SID103304585]
Effect on the antagonism of bicuculline-induced tonic-extensor convulsions (B) [AID113642, Type: Literature]
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3
[SID103304585]
Effect on the antagonism of nicotine-induced death (D) [AID113644, Type: Literature]
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4
[SID103304585]
Effect on the antagonism of nicotine-induced tonic-extensor convulsions (TE) in mice [AID113646, Type: Literature]
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5
[SID103304585]
Effect on the antagonism of oxotremorine-induced hypothermia (OX) [AID113648, Type: Literature]
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6
[SID103304585]
Effect on the antagonism of pentylenetetrazole-induced clonic convulsions (P) [AID113650, Type: Literature]
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7
[SID103304585]
Effect of test compound on the potentiation of apomorphine-induced gnawing (AG) in aggregated mice [AID113652, Type: Literature]
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8
[SID103304585]
Volume of distribution at steady state in human after iv administration [AID540209, Type: Literature]
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9
[SID103304585]
Clearance in human after iv administration [AID540210, Type: Literature]
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10
[SID103304585]
Fraction unbound in human after iv administration [AID540211, Type: Literature]
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11
[SID103304585]
Mean residence time in human after iv administration [AID540212, Type: Literature]
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12
[SID103304585]
Half life in human after iv administration [AID540213, Type: Literature]
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13
[SID103304585]
Renal clearance in human [AID444053, Type: Literature]
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14
[SID103304585]
Oral bioavailability in human [AID444054, Type: Literature]
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15
[SID103304585]
Fraction absorbed in human [AID444055, Type: Literature]
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16
[SID103304585]
Fraction escaping gut-wall elimination in human [AID444056, Type: Literature]
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17
[SID103304585]
Fraction escaping hepatic elimination in human [AID444057, Type: Literature]
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18
[SID103304585]
Volume of distribution at steady state in human [AID444058, Type: Literature]
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19
[SID103304585]
Virtual screen for compounds with anticonvulsant activity [AID227699, Type: Literature]
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20
[SID103304585]
Total body clearance in human [AID425652, Type: Literature]
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21
[SID103304585]
Renal clearance in human [AID425653, Type: Literature]
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22
[SID103304585]
Fraction unbound in human plasma [AID444050, Type: Literature]
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23
[SID103304585]
Total clearance in human [AID444051, Type: Literature]
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24
[SID103304585]
Hepatic clearance in human [AID444052, Type: Literature]
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25
[SID103304585]
Tested for antagonism of oxotremorine hypothermia (OX) in mice [AID114395, Type: Literature]
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26
[SID103304585]
Tested for antagonism of pentylenetetrazole-induced clonic convulsions (P) in mice [AID114396, Type: Literature]
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27
[SID103304585]
Tested for potentiation of gamma-butyrolactone induced sleep (gamma-B) in mice [AID114561, Type: Literature]
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28
[SID103304585]
Tested for potentiation of yohimbine toxicity in aggregated mice(Y) [AID114562, Type: Literature]
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29
[SID103304585]
Prolongation of hypoxic survival time (HS) in mice [AID114563, Type: Literature]
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30
[SID103304585]
Tested for stereotyped gnawing and licking behavior of mice pretreated with apomorphine (AG) [AID114565, Type: Literature]
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31
[SID103304585]
Effect on the potentiation of gamma-butyrolactone-induced sleep (gamma-B) [AID113655, Type: Literature]
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32
[SID103304585]
Effect on the potentiation of yohimbine-induced toxicity (Y) in aggregated mice [AID113656, Type: Literature]
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33
[SID103304585]
Effect on the prolongation of hypoxic survival time (HS) [AID113658, Type: Literature]
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34
[SID103304585]
Tested for antagonism of bicuculline-induced tonic-extensor convulsions (B) in mice [AID114392, Type: Literature]
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35
[SID103304585]
Tested for antagonism of nicotine-induced death (D) in mice [AID114393, Type: Literature]
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36
[SID103304585]
Tested for antagonism of nicotine-induced tonic extensor convulsions (TE) in mice [AID114394, Type: Literature]
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