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Lidocaine (CID 3676) - Compound BioActivity Data
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BioActivity Outcomes:
Active(31)
 
 
Inactive(1288)
 
 
Inconclusive(50)
 
 
Unspecified(613)
 
 
Top Targets:
7TM GPCR Srx(48)
 
 
 
 
7TM GPCR Srsx(37)
 
 
 
p450(28)
 
 
 
 
Na trans asso..(25)
 
 
 
Tryp SPc(17)
 
 
 
BioAssay Types:
Confirmatory(714)
 
 
 
 
Screening(539)
 
 
 
Literature(456)
 
 
 
 
 
Summary(24)
 
 
 
BioActivity Types:
Potency(502)
 
 
 
 
IC50(192)
 
 
 
 
EC50(11)
 
 
 
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 1564    Data Row: 1982   Total Pages: 100   Display: Page     
Sort: [Click the result table header to sort]
#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID103169867]
EC50 0.017Negative inotropic activity against potassium-induced contraction in guinea pig left atrium assessed as decrease in developed tension [AID491141, Type: Literature]
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2
[SID103169867]
EC50 0.017Negative inotropic activity in guinea pig left atria assessed as decrease of 1 Hz current-induced developed tension [AID655940, Type: Literature]
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3
[SID103169867]
EC50 0.017Negative inotropic activity assessed as decrease in developed tension in isolated guinea pig left atrium [AID275639, Type: Literature]
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4
[SID103169867]
Relative effect on slowing of ventricular tachycardia in dogs;slowing of VT present [AID60348, Type: Literature]
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5
[SID855682]
Aqueous Solubility from MLSMR Stock Solutions [AID1996, Type: other]
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6
[SID855682]
qHTS Assay for Spectroscopic Profiling in 4-MU Spectral Region [AID589, Type: other]
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7
[SID855682]
qHTS Assay for Spectroscopic Profiling in A350 Spectral Region [AID590, Type: other]
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8
[SID11110520]
NINDS Anticonvulsant Data (Qualitative) [AID423, Type: other]
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9
[SID11110520]
NINDS Anticonvulsant Data (Quantitative) [AID424, Type: other]
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10
[SID103169867]
Inhibition of yeast prion protein Sup35 infection of PSI yeast spheroplast cells at 200 uM [AID497664, Type: Literature]
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11
[SID103169867]
Relative effect on exacerbation of ventricular tachycardia in dogs; Exacerbation of VT present [AID60332, Type: Literature]
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12
[SID103169867]
Sodium channel alpha subunit blocker [AID742738, Type: Literature]Sodium channel protein type 1 subunit alpha [gi:12644229]
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13
[SID103169867]
Sodium channel alpha subunit blocker [AID742738, Type: Literature]Sodium channel protein type 1 subunit alpha [gi:12644229]
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14
[SID103169867]
Sodium channel alpha subunit blocker [AID742738, Type: Literature]Sodium channel protein type 2 subunit alpha [gi:25014053]
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15
[SID103169867]
Sodium channel alpha subunit blocker [AID742738, Type: Literature]Sodium channel protein type 2 subunit alpha [gi:25014053]
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16
[SID103169867]
Sodium channel alpha subunit blocker [AID742738, Type: Literature]Sodium channel protein type 3 subunit alpha [gi:25014054]
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17
[SID103169867]
Sodium channel alpha subunit blocker [AID742738, Type: Literature]Sodium channel protein type 3 subunit alpha [gi:25014054]
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18
[SID103169867]
Sodium channel alpha subunit blocker [AID742738, Type: Literature]Sodium channel protein type 8 subunit alpha [gi:34098756]
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19
[SID103169867]
Sodium channel alpha subunit blocker [AID742738, Type: Literature]Sodium channel protein type 8 subunit alpha [gi:34098756]
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20
[SID103169867]
Sodium channel alpha subunit blocker [AID742738, Type: Literature]Sodium channel protein type 11 subunit alpha [gi:124053649]
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