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2-(3-methoxyphenyl)-N,N-dimethylquinazolin-4-amine (CID 3233811) - Compound BioActivity Data
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BioActivity Outcomes:
Active(14)
 
 
Inactive(67)
 
 
Inconclusive(19)
 
 
Unspecified(1)
 
 
Top Targets:
p450(9)
 
 
 
 
HSD10-like SD..(4)
 
 
 
PKc CLK1 4(3)
 
 
ampC(2)
 
 
CASc(2)
 
 
BioAssay Types:
Confirmatory(87)
 
 
 
 
Screening(1)
 
 
BioActivity Types:
Potency(61)
 
 
 
 
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 90    Data Row: 101   Total Pages: 6   Display: Page     
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#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID4238702]
Potency 5.0119qHTS Assay for Inhibitors and Substrates of Cytochrome P450 3A4 [AID884, Type: confirmatory]cytochrome P450 3A4 isoform 1 [Homo sapiens] [gi:13435386]
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2
[SID4238702]
Potency 7.0795qHTS Assay for Inhibitors of CDC-like Kinase 4 (ADP-Glo Assay) [AID1771, Type: confirmatory]dual specificity protein kinase CLK4 [Homo sapiens] [gi:10190706]
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3
[SID4238702]
Potency 11.2202qHTS Assay for Inhibitors of CDC-like Kinase 4 (ADP-FP Assay) [AID1795, Type: confirmatory]dual specificity protein kinase CLK4 [Homo sapiens] [gi:10190706]
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4
[SID4238702]
Potency 11.2202qHTS Assay for Inhibitors of CDC-like Kinase 4 (Kinase-Glo Assay) [AID1770, Type: confirmatory]dual specificity protein kinase CLK4 [Homo sapiens] [gi:10190706]
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5
[SID4238702]
Potency 12.5893qHTS Assay for Inhibitors and Substrates of Cytochrome P450 2D6 [AID891, Type: confirmatory]cytochrome P450 2D6 isoform 1 [Homo sapiens] [gi:40805836]
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6
[SID4238702]
Potency 19.9526qHTS Assay for Inhibitors and Substrates of Cytochrome P450 2C19 [AID899, Type: confirmatory]cytochrome P450 2C19 precursor [Homo sapiens] [gi:4503219]
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7
[SID4238702]
Potency 25.1189qHTS Assay for Inhibitors of HADH2 (Hydroxyacyl-Coenzyme A Dehydrogenase, Type II) [AID886, Type: confirmatory]Chain A, The Structure Of Wild-Type Human Hadh2 (17beta-Hydroxysteroid Dehydrogenase Type 10) Bound To Nad+ At 1.2 A [gi:122921310]
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8
[SID4238702]
Potency 25.1189qHTS Assay for Inhibitors of HADH2 (Hydroxyacyl-Coenzyme A Dehydrogenase, Type II) [AID886, Type: confirmatory]Chain B, The Structure Of Wild-Type Human Hadh2 (17beta-Hydroxysteroid Dehydrogenase Type 10) Bound To Nad+ At 1.2 A [gi:122921311]
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9
[SID4238702]
Potency 56.2341Inhibitors of the vitamin D receptor (VDR): qHTS [AID504847, Type: confirmatory]vitamin D3 receptor isoform VDRA [Homo sapiens] [gi:63054845]
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10
[SID4238702]
Cytochrome panel assay with activity outcomes [AID1851_2, Type: other]cytochrome P450 2D6 isoform 2 [Homo sapiens] [gi:68509921]
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11
[SID4238702]
Cytochrome panel assay with activity outcomes [AID1851_1, Type: other]cytochrome P450 2C19 precursor [Homo sapiens] [gi:4503219]
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12
[SID4238702]
p450-cyp1a2 [AID410, Type: confirmatory]cytochrome P450 1A2 [Homo sapiens] [gi:73915100]
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13
[SID4238702]
Cytochrome panel assay with activity outcomes [AID1851_4, Type: other]cytochrome P450 1A2 [Homo sapiens] [gi:73915100]
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14
[SID4238702]
Cytochrome panel assay with activity outcomes [AID1851_3, Type: other]cytochrome P450 3A4 isoform 1 [Homo sapiens] [gi:13435386]
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15
[SID4238702]
Cytochrome panel assay with activity outcomes [AID1851, Type: other]
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16
[SID4238702]
Potency 0.7943qHTS Assay for Inhibitors and Substrates of Cytochrome P450 2C9 [AID883, Type: confirmatory]cytochrome P450 2C9 precursor [Homo sapiens] [gi:13699818]
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17
[SID4238702]
Potency 5.0119qHTS Assay for Activators of Cytochrome P450 3A4 [AID885, Type: confirmatory]cytochrome P450 3A4 isoform 1 [Homo sapiens] [gi:13435386]
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18
[SID4238702]
Potency qHTS for Inducers of the Endoplasmic Reticulum Stress Response (ERSR) in Human Glioma: qHTS [AID602332, Type: confirmatory]heat shock 70kDa protein 5 (glucose-regulated protein, 78kDa) [Homo sapiens] [gi:168984549]
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19
[SID4238702]
qHTS Assay for Inhibitors of RGS12 GoLoco Motif Activity (Red Fluorophore) [AID880, Type: confirmatory]guanine nucleotide-binding protein G(i) subunit alpha-1 isoform 1 [Homo sapiens] [gi:33946324]
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20
[SID4238702]
qHTS Assay for Inhibitors of Fructose-1,6-bisphosphate Aldolase from Giardia Lamblia: Coupling assay counterscreen [AID2472, Type: screening]glyceraldehyde-3-phosphate dehydrogenase isoform 1 [Homo sapiens] [gi:7669492]
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