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coumarin (CID 323) - Compound BioActivity Data
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BioActivity Outcomes:
Active(49)
 
 
Inactive(1452)
 
 
Inconclusive(60)
 
 
Unspecified(1481)
 
 
Top Targets:
NR LBD PPAR(45)
 
 
 
7TM GPCR Srx(40)
 
 
 
7TM GPCR Srsx(38)
 
 
 
NR LBD ER(29)
 
 
 
 
 
NR LBD AR(28)
 
 
 
 
BioAssay Types:
Confirmatory(865)
 
 
 
 
 
Screening(531)
 
 
 
 
Literature(272)
 
 
 
 
 
Summary(72)
 
 
 
BioActivity Types:
Potency(655)
 
 
 
 
 
IC50(174)
 
 
 
 
Ki(50)
 
 
 
EC50(8)
 
 
 
AC50(2)
 
 
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 2536    Data Row: 3042   Total Pages: 153   Display: Page     
Sort: [Click the result table header to sort]
#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID103164854]
Ki 0.048Inhibition of human carbonic anhydrase 14 by stopped flow CO2 hydration assay [AID444782, Type: Literature]Carbonic anhydrase 14 [gi:8928036]
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2
[SID103164854]
Km 0.64Michaelis-Menten constant of compound against mouse cytochrome P450 2A5 enzyme [AID239733, Type: Literature]
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3
[SID103164854]
Km 0.74Michaelis-Menten constant of compound against human cytochrome P450 2A6 enzyme [AID239732, Type: Literature]Cytochrome P450 2A6 [gi:308153612]
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4
[SID103164854]
Ki 2Inhibition of human carbonic anhydrase 6 by stopped flow CO2 hydration assay [AID444777, Type: Literature]Carbonic anhydrase 6 [gi:116241278]
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5
[SID103164854]
Ki 3.1Inhibition of human CA1 pre-incubated for 15 mins to 24 hrs measured after 6 hrs by phenol red-based stopped-flow CO2 hydrase assay [AID639299, Type: Literature]Carbonic anhydrase 1 [gi:115449]
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6
[SID103164854]
Ki 3.1Inhibition of human full-length cytosolic CA1 after 6 hrs by stopped flow CO2 hydration assay [AID641823, Type: Literature]Carbonic anhydrase 1 [gi:115449]
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7
[SID103164854]
Ki 3.1Inhibition of human recombinant carbonic anhydrase 1 preincubated for 15 mins to 72 hrs measured after 6 hrs by stopped flow CO2 hydration method [AID649891, Type: Literature]Carbonic anhydrase 1 [gi:115449]
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8
[SID103164854]
Ki 3.1Inhibition of full length human recombinant CA1 cytosolic isoform after 6 hrs by stopped-flow CO2 hydration method [AID727279, Type: Literature]Carbonic anhydrase 1 [gi:115449]
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9
[SID103164854]
Ki 3.1Inhibition of human carbonic anhydrase 1 preincubated for 6 hrs by CO2 hydration stopped-flow assay [AID729563, Type: Literature]Carbonic anhydrase 1 [gi:115449]
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10
[SID103164854]
Ki 3.1Inhibition of human carbonic anhydrase 1 after 6 hrs by stop-flow CO2 hydration assay [AID650662, Type: Literature]Carbonic anhydrase 1 [gi:115449]
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11
[SID103164854]
Ki 3.1Inhibition of full length human CA1 cytosolic isoform by stopped-flow CO2 hydration method [AID539679, Type: Literature]Carbonic anhydrase 1 [gi:115449]
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12
[SID103164854]
Ki 3.1Inhibition of human carbonic anhydrase 1 by stopped flow CO2 hydration assay [AID444771, Type: Literature]Carbonic anhydrase 1 [gi:115449]
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13
[SID103164854]
Ki 3.3Inhibition of human carbonic anhydrase 7 by stopped flow CO2 hydration assay [AID444778, Type: Literature]Carbonic anhydrase 7 [gi:1168744]
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14
[SID103164854]
Ki 5.2Inhibition of human carbonic anhydrase 5B by stopped flow CO2 hydration assay [AID444776, Type: Literature]Carbonic anhydrase 5B, mitochondrial [gi:8928041]
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15
[SID103164854]
Ki 5.6Inhibition of human carbonic anhydrase 3 by stopped flow CO2 hydration assay [AID444773, Type: Literature]Carbonic anhydrase 3 [gi:134047703]
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16
[SID103164854]
Ki 6.8Inhibition of human carbonic anhydrase 4 by stopped flow CO2 hydration assay [AID444774, Type: Literature]Carbonic anhydrase 4 [gi:115465]
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17
[SID103164854]
Ki 8.9Inhibition of human carbonic anhydrase 12 by stopped flow CO2 hydration assay [AID444780, Type: Literature]Carbonic anhydrase 12 [gi:5915866]
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18
[SID103164854]
Ki 9.1Inhibition of human carbonic anhydrase 9 by stopped flow CO2 hydration assay [AID444779, Type: Literature]Carbonic anhydrase 9 [gi:83300925]
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19
[SID103164854]
Ki 9.2Inhibition of mouse carbonic anhydrase 13 by stopped flow CO2 hydration assay [AID444781, Type: Literature]Carbonic anhydrase 13 [gi:30580372]
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20
[SID103164854]
Ki 9.2Inhibition of full length human CA2 cytosolic isoform by stopped-flow CO2 hydration method [AID539680, Type: Literature]Carbonic anhydrase 2 [gi:115456]
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